Description

Elopiprazole is a high-purity pharmaceutical intermediate and research chemical with significant importance in modern medicinal chemistry. Its primary value lies in its role as a key building block for the synthesis of novel therapeutic agents, particularly in the central nervous system (CNS) domain. This compound is essential for pharmaceutical R&D laboratories, contract manufacturing organizations (CMOs), and academic institutions engaged in drug discovery and process development.

Application

• Pharmaceutical Intermediate: Serves as a critical precursor in the synthesis of advanced active pharmaceutical ingredients (APIs) for neurological and psychiatric research.
• Drug Discovery & Development: Used as a reference standard and building block in medicinal chemistry programs targeting novel CNS pathways.
• Chemical Research: Employed in academic and industrial research to study structure-activity relationships (SAR) and develop new synthetic methodologies.
• Process Chemistry: Utilized for scaling up and optimizing synthetic routes in pilot plants and commercial manufacturing settings.
• Reference Standard: Acts as a high-purity analytical standard for quality control and method validation in analytical laboratories.

Basic Information

Product Name	Elopiprazole
CAS No.	115464-77-2
Molecular Formula	C21H24FN3O2S
Molecular Weight	401.50 g/mol
Synonyms	1-(4-Fluorophenyl)-4-[(6-methyl-2-pyridinyl)methyl]-1,2,3,6-tetrahydro-5-(methylsulfonyl)pyrrolo[3,4-c]pyrazole; Elopiprazole (USAN); UNII-9B6K5V3Y6I; 9B6K5V3Y6I; Pyrrolo[3,4-c]pyrazole-5(1H)-sulfonamide derivative; CNS Research Compound
EINECS	Contact for details

Quality Control

Our Elopiprazole is manufactured under strict quality management systems to ensure batch-to-batch consistency and high purity suitable for research and development applications. Each lot undergoes comprehensive analytical testing, including HPLC, NMR, and MS, to verify identity and purity. A detailed Certificate of Analysis (COA) is provided with every shipment, documenting all critical quality attributes.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry, and well-ventilated place at a controlled room temperature (15-25°C). Due to its hygroscopic (moisture-sensitive) nature, the container must be kept tightly sealed after each use to prevent degradation from atmospheric moisture. Keep away from incompatible materials.

Specification

Item	Specification
Appearance	White to off-white powder
Identification (IR)	Conforms to reference spectrum
Identification (HPLC)	Retention time matches reference standard
Assay (HPLC)	≥ 98.0%
Related Substances (HPLC)	Total impurities ≤ 2.0%
Water Content (KF)	≤ 0.5%
Residue on Ignition	≤ 0.1%

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.