Description

Rilmenidine is a highly selective imidazoline I1 receptor agonist, primarily recognized for its role in cardiovascular research and pharmaceutical development. This compound is valued for its specific mechanism of action, which makes it a critical intermediate and reference standard in the synthesis of antihypertensive agents. It is essential for pharmaceutical manufacturers, research institutions, and chemical suppliers serving the global life sciences sector. Rilmenidine CAS NO 54187-04-1 is supplied under stringent quality controls to ensure reliability for advanced applications.

Application

• Pharmaceutical Active Ingredient (API): Serves as the core active component in the formulation of antihypertensive medications.
• Biochemical Research: Used as a selective pharmacological tool to study imidazoline receptor pathways and central nervous system-mediated blood pressure regulation.
• Reference Standard: Employed in analytical laboratories for method development, validation, and quality control testing of drug substances and products.
• Chemical Synthesis: Acts as a key intermediate in the organic synthesis of more complex molecules targeting cardiovascular diseases.
• Preclinical & Clinical Studies: Utilized in animal models and clinical trials to investigate efficacy, pharmacokinetics, and safety profiles.

Basic Information

Product Name	Rilmenidine
CAS No.	54187-04-1
Molecular Formula	C10H17N3O2
Molecular Weight	211.26 g/mol
Synonyms	Rilmenidine; S 3341; S-3341; (N-Dicyclopropylmethyl)-4,5-dihydro-2-oxazolamine; 2-[(Dicyclopropylmethyl)amino]-4,5-dihydro-1,3-oxazole; Oxaminozoline; Tenaxum
EINECS	Contact for details

Quality Control

Our Rilmenidine is manufactured and tested to meet the high-purity standards required for pharmaceutical research and development. Each batch undergoes comprehensive analytical testing, including identification, assay, and impurity profiling, to ensure compliance with internal specifications and relevant pharmacopeial guidelines. A Certificate of Analysis (COA) detailing all test results is provided with every shipment to guarantee traceability and quality assurance.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry place at controlled room temperature (15-25°C). The product is light-sensitive and should be handled accordingly to maintain stability.

Specification

Item	Specification
Appearance	White to off-white crystalline powder
Identification (IR)	Conforms to reference spectrum
Identification (HPLC)	Retention time matches reference standard
Assay (HPLC)	≥ 98.5%
Related Substances (HPLC)	Total impurities ≤ 1.5% Any single impurity ≤ 0.5%
Residual Solvents (GC)	Complies with ICH Q3C guidelines
Loss on Drying	≤ 0.5%
Heavy Metals	≤ 20 ppm

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.