Description

Epertinib Hydrochloride CAS NO 2071195-74-7 is a highly potent and selective small molecule inhibitor targeting specific tyrosine kinases. This compound is of significant value in pharmaceutical research and development, particularly in the field of oncology. It is primarily needed by pharmaceutical manufacturers, biotechnology research firms, and academic institutions engaged in the discovery and synthesis of novel therapeutic agents for cancer treatment.

Application

• Pharmaceutical Intermediate: Serves as a critical active pharmaceutical ingredient (API) in the development of targeted cancer therapies.
• Oncology Research: Used as a reference standard and biochemical tool in preclinical studies to investigate kinase inhibition pathways.
• Drug Discovery & Development: A key compound for high-throughput screening and structure-activity relationship (SAR) studies in medicinal chemistry.
• Clinical Trial Material: Supplied under GMP guidelines for use in formulating investigational new drugs for clinical trials.
• Biochemical Assays: Employed in enzymatic assays to study potency, selectivity, and mechanism of action against specific kinase targets.

Basic Information

Item	Details
Product Name	Epertinib Hydrochloride
CAS No.	2071195-74-7
Molecular Formula	Contact for details
Molecular Weight	Contact for details
Synonyms	Epertinib HCl; Epertinib Hydrochloride Salt; TAS-119; TAS119; (R,E)-N-(7-Chloro-1-(1-(4-fluorophenyl)-1-hydroxypropan-2-yl)-1H-indazol-5-yl)-3-(2-methylpyrimidin-4-yl)acrylamide hydrochloride
EINECS	Contact for details

Quality Control

Our Epertinib Hydrochloride is manufactured under strict quality management systems. Each batch undergoes rigorous analytical testing, including HPLC for purity and identity confirmation, to ensure it meets the high standards required for pharmaceutical research. Certificates of Analysis (COA) detailing all test results are available upon request to support your quality assurance and regulatory documentation.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry place at a controlled room temperature (typically 15-25°C). Due to its hygroscopic nature, the container must be kept tightly sealed in a dry environment to prevent moisture absorption, which can affect stability and purity.

Specification

Item	Specification
Appearance	White to off-white powder
Identification (HPLC)	Conforms to reference standard
Identification (IR)	Conforms to structure
Assay (HPLC)	≥ 98.0%
Related Substances (HPLC)	Total impurities ≤ 2.0%
Water Content (KF)	≤ 1.0%
Residue on Ignition	≤ 0.1%

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.