Description

Tk216 CAS NO 1903783-48-1 is a high-purity, small molecule compound of significant interest in advanced pharmaceutical research and development. This compound serves as a critical intermediate or active pharmaceutical ingredient (API) for the synthesis of novel therapeutic agents. It is primarily utilized by research institutions and pharmaceutical companies engaged in oncology, immunology, and other life science fields requiring precise chemical building blocks.

Application

• Pharmaceutical Intermediate: A key building block in the multi-step synthesis of targeted drug candidates, particularly in oncology research.
• Biochemical Research: Used as a reference standard or probe molecule in enzymatic assays and cellular pathway studies.
• Preclinical Development: Serves as a critical material for pharmacokinetic (PK), pharmacodynamic (PD), and toxicology studies during drug discovery.
• Proteolysis-Targeting Chimera (PROTAC) Development: Potential application as a warhead or linker component in the design of novel targeted protein degraders.
• Kinase Inhibitor Research: Acts as a scaffold or precursor for the development of selective kinase inhibitors.
• Chemical Biology: Employed in the study of protein-ligand interactions and the identification of novel biological targets.

Basic Information

Product Name	Tk216
CAS No.	1903783-48-1
Molecular Formula	Contact for details
Molecular Weight	Contact for details
Synonyms	TK-216; (S,E)-N-(1-(4-(N-(2-(Dimethylamino)ethyl)sulfamoyl)phenyl)ethyl)-6-(4-fluorostyryl)imidazo[1,2-a]pyridine-3-carboxamide; 1903783-48-1; UNII-1V5P8C0T9M; 1V5P8C0T9M; Tk 216; Tk-216 (EZH2 inhibitor); BDBM50389365; HY-101526; ZINC000006714007; AKOS009456046; CS-0536130; FT-0717137; NS-00061367; A31227; SR-01000931073; Q27283015
EINECS	Contact for details

Quality Control

Our Tk216 is manufactured under strict quality management systems. Each batch undergoes rigorous analytical testing, including HPLC, NMR, and MS, to ensure identity, purity, and consistency. Certificates of Analysis (COA) with detailed chromatographic data are provided for every shipment, supporting your regulatory and research documentation needs.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry place at a controlled room temperature (15-25°C). Due to its hygroscopic (moisture-sensitive) nature, the container must be kept tightly sealed in a dry environment to prevent degradation. For long-term storage, consider using desiccants.

Specification

Item	Specification
Appearance	White to off-white solid
Identification (HPLC)	Conforms
Identification (MS)	Conforms
Purity (HPLC)	≥ 98.0%
Water Content (KF)	≤ 1.0%
Residual Solvents (GC)	Complies with ICH Q3C

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.