Description

2-(Morpholin-4-Yl)Pyridin-3-Ylboronic Acid is a specialized boronic acid derivative that serves as a crucial building block in modern synthetic chemistry. Its core value lies in enabling the efficient construction of complex molecules through reliable cross-coupling reactions. This high-purity intermediate is essential for researchers and manufacturers in the pharmaceutical and agrochemical industries developing new active ingredients.

Application

• Pharmaceutical Intermediate: A key precursor in Suzuki-Miyaura cross-coupling reactions for synthesizing novel drug candidates, particularly in kinase inhibitor and CNS-active compound research.
• Agrochemical Synthesis: Used in the development of advanced herbicides, fungicides, and insecticides that require complex heterocyclic architectures.
• Material Science Research: Employed in the synthesis of organic electronic materials, such as ligands for OLEDs and conductive polymers.
• Chemical Biology Probes: Facilitates the creation of tagged molecules and bioconjugates for studying biological pathways and protein interactions.
• Catalyst Ligand Development: Acts as a starting material for synthesizing novel bidentate ligands used in homogeneous catalysis.
• Custom Synthesis & Contract Manufacturing: Supplied to CDMOs for the production of bespoke compounds under cGMP conditions for clinical trials.

Basic Information

Product Name	2-(Morpholin-4-Yl)Pyridin-3-Ylboronic Acid
CAS No.	1218790-86-3
Molecular Formula	C9H13BN2O3
Molecular Weight	208.03 g/mol
Synonyms	2-(4-Morpholinyl)-3-pyridineboronic acid; 3-Borono-2-(morpholin-4-yl)pyridine; 2-Morpholin-4-ylpyridine-3-boronic acid; [2-(Morpholin-4-yl)pyridin-3-yl]boronic acid; 1218790-86-3; 2-(N-Morpholino)pyridine-3-boronic acid; 3-Pyridineboronic acid, 2-(4-morpholinyl)-
EINECS	Contact for details

Quality Control

Our 2-(Morpholin-4-Yl)Pyridin-3-Ylboronic Acid is manufactured under strict quality management systems. Each batch undergoes rigorous analytical testing, including HPLC for purity and NMR for structural confirmation, to ensure compliance with stringent industry standards. Comprehensive Certificates of Analysis (COA) detailing purity, identity, and impurity profiles are available upon request to support your regulatory and R&D needs.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry, and well-ventilated place at a controlled room temperature (15-25°C). Due to its hygroscopic nature, the container must be kept tightly sealed under an inert atmosphere (e.g., nitrogen or argon) after opening to prevent moisture absorption and decomposition.

Specification

Item	Specification
Appearance	White to off-white powder
Identification (IR)	Conforms to structure
Purity (HPLC)	≥ 97.0%
Water Content (KF)	≤ 0.5%

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.