Description

4-[(1,3-Dihydro-1-Hydroxy-2,1-Benzoxaborol-5-Yl)Oxy]-Benzamide is a specialized benzoxaborole derivative, a class of compounds recognized for their unique biological activity and utility in advanced chemical synthesis. This compound matters as a high-value pharmaceutical intermediate and research chemical, offering a critical building block for the development of novel therapeutic agents. It is primarily needed by R&D laboratories and pharmaceutical manufacturers focused on antifungal, antibacterial, and anti-inflammatory drug discovery programs.

Application

• Pharmaceutical Intermediate: Serves as a key precursor in the synthesis of novel benzoxaborole-based active pharmaceutical ingredients (APIs).
• Biochemical Research: Used as a probe or inhibitor in enzymatic studies and target validation for infectious diseases.
• Antifungal Agent Development: Exploited for its potential mechanism of action against fungal pathogens in preclinical research.
• Antibacterial Compound Synthesis: Incorporated into molecular structures designed to combat antibiotic-resistant bacteria.
• Boronic Acid Derivative Chemistry: Utilized in Suzuki-Miyaura cross-coupling reactions and other catalytic processes due to its boronate ester functionality.
• Medicinal Chemistry Libraries: A valuable scaffold for constructing diverse compound libraries for high-throughput screening.

Basic Information

Product Name	4-[(1,3-Dihydro-1-Hydroxy-2,1-Benzoxaborol-5-Yl)Oxy]-Benzamide
CAS No.	1187188-59-5
Molecular Formula	C14H12BNO4
Molecular Weight	269.06 g/mol
Synonyms	5-(4-Carbamoylphenoxy)-2,1-benzoxaborol-1(3H)-ol; 4-((1-Hydroxy-1,3-dihydrobenzo[c][1,2]oxaborol-5-yl)oxy)benzamide; Benzamide, 4-[(1,3-dihydro-1-hydroxy-2,1-benzoxaborol-5-yl)oxy]-; AN-465/43403029; BCP31989; ZB1606; AKOS025310065; 1-Hydroxy-5-(4-carbamoylphenoxy)-1,3-dihydro-2,1-benzoxaborole
EINECS	Contact for details

Quality Control

Our 4-[(1,3-Dihydro-1-Hydroxy-2,1-Benzoxaborol-5-Yl)Oxy]-Benzamide is manufactured under a strict quality management system. Each batch undergoes rigorous analytical testing, including HPLC, NMR, and MS, to ensure identity, purity, and consistency. Certificates of Analysis (COA) detailing all specifications are provided and available upon request to support your quality assurance and regulatory needs.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry, and well-ventilated area at a controlled room temperature (15-25°C). Due to its hygroscopic (moisture-sensitive) nature, the container must be kept tightly sealed after each use to prevent degradation from atmospheric moisture.

Specification

Item	Specification
Appearance	White to off-white powder
Identification (IR)	Conforms to structure
Identification (NMR)	Conforms to structure
Purity (HPLC)	≥ 97.0%
Water Content (KF)	≤ 1.0%
Residue on Ignition	≤ 0.5%
Heavy Metals	≤ 20 ppm

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.