Cholinergic Drugs

Cholinergic Drugs

Cholinergic drugs modulate the cholinergic neurotransmitter system by either enhancing acetylcholine activity or inhibiting its breakdown. This category includes direct agonists, indirect cholinesterase inhibitors, and agents that augment cholinergic tone in the central or peripheral nervous system. These drugs are widely used in Alzheimer’s disease, myasthenia gravis, glaucoma, gastrointestinal motility disorders, and certain types of poisoning. Their mechanisms involve stimulating muscarinic or nicotinic receptors, prolonging acetylcholine availability, or restoring synaptic transmission in neuromuscular junctions. While beneficial, cholinergic drugs may cause side effects such as bradycardia, excessive secretions, gastrointestinal discomfort, and cholinergic crisis, necessitating careful dosing and monitoring. They remain crucial in both neurological and autonomic therapeutics.

Tacrine Hydrochloride CAS NO 1684-40-8

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CAS No.:1684-40-8

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Content:99.90%

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Propionylcholine p-Toluenesulfonate CAS NO 1866-13-3

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CAS No.:1866-13-3

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Galantamine Hydrobromide CAS NO 1953-04-4

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CAS No.:1953-04-4

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Deptropine Methobromide CAS NO 10139-98-7

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CAS No.:10139-98-7

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n-Methylcarbamylcholine CAS NO 14721-69-8

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CAS No.:14721-69-8

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Dimethylcarbamylcholine CAS NO 14721-70-1

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CAS No.:14721-70-1

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Methylcarbamylcholine Chloride Nicotinic Agonist CAS NO 14721-76-7

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CAS No.:14721-76-7

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Tofenacin CAS NO 15301-93-6

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CAS No.:15301-93-6

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