Description

1-(2-Boronophenylsulfonyl)Piperidine is a specialized organoboron building block featuring a sulfonyl linker, which is critical for modern cross-coupling reactions in pharmaceutical and agrochemical research. This compound matters because it provides a unique handle for Suzuki-Miyaura coupling, enabling the efficient construction of complex biaryl and heterobiaryl structures central to drug discovery. Research and development teams in the pharmaceutical, agrochemical, and advanced materials sectors need this high-purity intermediate to accelerate their synthetic programs and develop novel active ingredients.

Application

• Pharmaceutical Intermediate: A key synthon in the synthesis of active pharmaceutical ingredients (APIs) via Suzuki-Miyaura cross-coupling reactions.
• Agrochemical Research: Used in the development of novel herbicides, fungicides, and insecticides requiring complex boron-containing scaffolds.
• Material Science: Serves as a precursor for creating organic electronic materials, such as those used in OLEDs and sensors.
• Chemical Biology: Employed as a probe or linker in bioconjugation chemistry and proteolysis-targeting chimera (PROTAC) development.
• Catalyst Ligand Synthesis: Acts as a building block for constructing sophisticated ligands used in homogeneous catalysis.
• Academic & Contract Research: Essential for methodological studies in organic synthesis and medicinal chemistry within R&D laboratories.

Basic Information

Product Name	1-(2-Boronophenylsulfonyl)Piperidine
CAS No.	957034-87-6
Molecular Formula	C11H16BNO4S
Molecular Weight	269.13 g/mol
Synonyms	2-(Piperidine-1-sulfonyl)phenylboronic acid; 1-[(2-Boronophenyl)sulfonyl]piperidine; Piperidine, 1-[(2-boronophenyl)sulfonyl]-; 2-(1-Piperidinesulfonyl)benzeneboronic acid; 1-(2-Boronobenzene-1-sulfonyl)piperidine; B-(2-((Piperidin-1-yl)sulfonyl)phenyl)boronic acid; 2-(Piperidin-1-ylsulfonyl)phenylboronic acid
EINECS	Contact for details

Quality Control

Our 1-(2-Boronophenylsulfonyl)Piperidine is manufactured under strict quality management systems to ensure batch-to-batch consistency and high purity for research and development applications. Each lot undergoes comprehensive analytical testing, including HPLC, NMR, and elemental analysis. A Certificate of Analysis (COA) detailing purity, identity, and impurity profiles is provided with every shipment to support your quality assurance protocols.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry, and well-ventilated place at a controlled room temperature (15-25°C). Due to its hygroscopic (moisture-sensitive) nature, the container must be kept sealed under an inert atmosphere (e.g., nitrogen or argon) after opening to prevent degradation.

Specification

Item	Specification
Appearance	White to off-white powder
Identification (IR)	Conforms to structure
Purity (HPLC)	≥ 97.0%
Water Content (KF)	≤ 1.0%
Heavy Metals	≤ 20 ppm

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.