Description

[2-(2-Methylmorpholin-4-Yl)Pyridin-4-Yl]Methanamine is a high-purity, advanced pharmaceutical intermediate featuring a unique heterocyclic structure combining pyridine and morpholine motifs. This compound is critical for medicinal chemistry research and development, particularly in the synthesis of targeted small molecule therapeutics. It is primarily sought after by pharmaceutical R&D laboratories and fine chemical manufacturers engaged in developing novel active pharmaceutical ingredients (APIs) for central nervous system (CNS) and other therapeutic areas.

Application

• Pharmaceutical Intermediate: A key building block in the synthesis of novel drug candidates, particularly those targeting neurological and psychiatric disorders.
• Medicinal Chemistry Research: Used in structure-activity relationship (SAR) studies and lead optimization programs due to its privileged scaffold.
• API Development: Serves as a critical precursor in the multi-step synthesis of complex Active Pharmaceutical Ingredients (APIs).
• Chemical Biology Probes: Utilized in the development of tool compounds and probes for studying biological pathways and target validation.
• Contract Research & Manufacturing (CRO/CMO): Supplied to organizations specializing in custom synthesis and process development for the pharmaceutical industry.
• Academic Research: Employed in university and institutional labs for exploratory synthetic chemistry and drug discovery projects.

Basic Information

Product Name	[2-(2-Methylmorpholin-4-Yl)Pyridin-4-Yl]Methanamine
CAS No.	953901-77-4
Molecular Formula	C11H17N3O
Molecular Weight	207.27 g/mol
Synonyms	4-(Aminomethyl)-2-(2-methylmorpholino)pyridine; 2-(2-Methylmorpholin-4-yl)pyridin-4-ylmethanamine; 4-Pyridinemethanamine, 2-(2-methyl-4-morpholinyl)-; (2-(2-Methylmorpholino)pyridin-4-yl)methanamine; 953901-77-4; UNII-9V3F6S8Q4K; 2-(2-Methylmorpholin-4-yl)pyridin-4-amine (Note: This is a common misnomer, the correct structure has an aminomethyl group)
EINECS	Contact for details

Quality Control

Our [2-(2-Methylmorpholin-4-Yl)Pyridin-4-Yl]Methanamine is manufactured under strict quality management systems. Each batch undergoes comprehensive analytical testing, including HPLC for purity, NMR and MS for structural confirmation, and residual solvent analysis, to ensure it meets the stringent requirements of pharmaceutical development. Certificates of Analysis (COA) with full traceability are provided with every shipment.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry, and well-ventilated place at a controlled room temperature (15-25°C). Due to its hygroscopic nature, the container must be kept tightly sealed to prevent moisture absorption, which may affect stability and handling properties. Keep away from incompatible materials.

Specification

Item	Specification
Appearance	White to off-white solid
Identification (HPLC)	Conforms to reference standard
Identification (NMR)	Conforms to structure
Purity (HPLC)	≥ 98.0%
Water Content (KF)	≤ 0.5%
Residual Solvents (GC)	Meets ICH Q3C guidelines

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.