Description

Benzyl 3-(Methoxy(Methyl)Carbamoyl)Azetidine-1-Carboxylate is a high-purity, advanced pharmaceutical intermediate with a complex heterocyclic structure. This compound is of significant value in modern organic synthesis, particularly for constructing novel bioactive molecules and peptidomimetics. It is primarily needed by research institutions and manufacturers in the pharmaceutical and agrochemical industries for the development of new active ingredients.

Application

• Pharmaceutical Intermediate: A key building block in the synthesis of novel drug candidates, particularly those targeting protease enzymes or requiring constrained azetidine scaffolds.
• Peptidomimetic Research: Used to create conformationally restricted peptide analogs for enhanced metabolic stability and receptor selectivity in drug discovery programs.
• Agrochemical Synthesis: Serves as a precursor in the development of new generation herbicides and fungicides with specific modes of action.
• Chemical Biology Probes: Employed in the design and synthesis of activity-based probes (ABPs) for studying enzyme function and target engagement.
• Custom Synthesis & Contract Manufacturing: Supplied to CDMOs (Contract Development and Manufacturing Organizations) for custom synthesis projects requiring specialized heterocyclic chemistry.
• Academic & R&D: Utilized in university and institutional research laboratories for methodological development in organic and medicinal chemistry.

Basic Information

Product Name	Benzyl 3-(Methoxy(Methyl)Carbamoyl)Azetidine-1-Carboxylate
CAS No.	937049-10-0
Molecular Formula	C15H20N2O4
Molecular Weight	292.33 g/mol
Synonyms	1-[(Benzyloxy)carbonyl]-3-[(methoxy(methyl)amino)carbonyl]azetidine; Benzyl 3-[(Methoxy(methyl)carbamoyl)]azetidine-1-carboxylate; 1-CBz-3-(N-Methoxy-N-methylcarbamoyl)azetidine; Azetidine-1-carboxylic acid, 3-[(methoxy(methyl)amino)carbonyl]-, phenylmethyl ester; N-Methoxy-N-methyl-1-[(phenylmethoxy)carbonyl]-3-azetidinecarboxamide
EINECS	Contact for details

Quality Control

Our Benzyl 3-(Methoxy(Methyl)Carbamoyl)Azetidine-1-Carboxylate is manufactured under strict quality management systems. Each batch undergoes rigorous analytical testing, including HPLC for purity and identity confirmation, to ensure it meets the high standards required for pharmaceutical R&D. A comprehensive Certificate of Analysis (COA) detailing purity, assay, and impurity profiles is provided with every shipment and is available upon request.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry, and well-ventilated area at a controlled room temperature (typically 15-25°C). The product should be kept under an inert atmosphere if long-term storage is required to maintain optimal stability.

Specification

Item	Specification
Appearance	White to off-white solid
Identification (IR)	Conforms to structure
Purity (HPLC)	≥ 97.0%
Assay	≥ 95.0%
Water Content (KF)	≤ 0.5%
Residue on Ignition	≤ 0.1%

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.