Description

Boc-3-Amino-1-Carboxymethyl-Pyridin-2-One is a high-purity, protected heterocyclic building block essential for advanced organic synthesis. This compound is specifically engineered to facilitate the controlled introduction of functionalized pyridone moieties into complex molecular architectures. It is a critical intermediate for researchers and manufacturers in the pharmaceutical and agrochemical industries developing novel active ingredients.

Application

• Pharmaceutical Intermediate: Key building block for the synthesis of novel drug candidates, particularly in kinase inhibitor and antiviral research.
• Peptidomimetic Synthesis: Used to incorporate heterocyclic scaffolds that mimic peptide structures, enhancing metabolic stability and bioavailability.
• Agrochemical Development: Serves as a precursor in creating new herbicides and fungicides with targeted modes of action.
• Chemical Biology Probes: Utilized in the development of molecular probes and labeled compounds for studying biological pathways.
• Material Science Research: A precursor for specialty polymers and ligands used in catalysis and sensing applications.
• Custom Synthesis & Contract Manufacturing: Supplied to CDMOs for the production of bespoke compounds and development-scale batches.

Basic Information

Product Name	Boc-3-Amino-1-Carboxymethyl-Pyridin-2-One
CAS No.	882847-09-8
Molecular Formula	C12H16N2O5
Molecular Weight	268.27 g/mol
Synonyms	1-(Carboxymethyl)-3-amino-2-oxo-1,2-dihydropyridine-1-carboxylic acid tert-butyl ester; tert-Butyl 3-amino-1-carboxymethyl-2-oxo-1,2-dihydropyridine-1-carboxylate; Boc-3-Amino-1-CM-Pyridin-2-One; N-Boc-3-Amino-1-Carboxymethyl-2-pyridone; 3-Amino-1-(carboxymethyl)pyridin-2(1H)-one tert-butyl carbonate; 882847-09-8; Boc-protected 3-aminopyridone acetic acid
EINECS	Contact for details

Quality Control

Our Boc-3-Amino-1-Carboxymethyl-Pyridin-2-One is manufactured under strict quality management systems. Each batch undergoes rigorous analytical testing, including HPLC for purity and identity confirmation by NMR and IR spectroscopy, to ensure it meets the high standards required for research and development. A comprehensive Certificate of Analysis (COA) detailing all specifications is provided with every shipment.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry, and well-ventilated place at a controlled room temperature (15-25°C). Due to its hygroscopic (moisture-sensitive) nature, the container must be kept tightly sealed after opening to prevent degradation from atmospheric moisture.

Specification

Item	Specification
Appearance	White to off-white crystalline powder
Identification (IR)	Conforms to structure
Purity (HPLC)	≥ 98.0%
Water Content (KF)	≤ 0.5%
Residue on Ignition	≤ 0.1%
Heavy Metals (as Pb)	≤ 10 ppm

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.