Description

Telenzepine 2Hcl is a high-purity muscarinic acetylcholine receptor antagonist, specifically targeting the M1 subtype. This compound is of significant value for pharmacological research and development, particularly in the study of gastrointestinal and central nervous system disorders. It is primarily required by pharmaceutical R&D laboratories, academic research institutions, and fine chemical manufacturers engaged in neurochemical synthesis.

Application

• Pharmacological Research: A key reference standard and tool compound for studying muscarinic M1 receptor function and antagonism.
• Drug Discovery Programs: Used in high-throughput screening and lead optimization for developing new therapeutics targeting cholinergic pathways.
• Academic Neuroscience Studies: Fundamental research into the role of specific muscarinic receptor subtypes in diseases like Alzheimer's, peptic ulcers, and smooth muscle disorders.
• Biochemical Assay Development: Serves as a critical control and validation agent in developing in vitro receptor binding and functional assays.
• Fine Chemical Synthesis: An intermediate or building block for the synthesis of more complex, targeted receptor modulators.
• Preclinical Development: Used in animal model studies to investigate the efficacy and mechanism of action of anticholinergic agents.

Basic Information

Product Name	Telenzepine 2Hcl
CAS No.	80880-90-6
Molecular Formula	C₁₉H₂₂Cl₂N₄O₂
Molecular Weight	409.31 g/mol
Synonyms	Telenzepine Dihydrochloride; 3,11-Dihydro-9-acridinyl-5H-pyrido[2,3-b][1,4]benzodiazepin-5-one Dihydrochloride; 9-Acridinyl-3,11-dihydro-5H-pyrido[2,3-b][1,4]benzodiazepin-5-one Dihydrochloride; Telenzepine HCl; LS 198-641; LS 198641
EINECS	Contact for details

Quality Control

Our Telenzepine 2Hcl is manufactured under strict quality management systems. Each batch undergoes rigorous analytical testing, including HPLC for purity and identity confirmation via spectroscopic methods, to ensure it meets the high standards required for research applications. A comprehensive Certificate of Analysis (COA) detailing purity, assay, and impurity profiles is provided with every shipment.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry place at a controlled room temperature (15-25°C). This product is hygroscopic (moisture-sensitive) and must be kept in a desiccated environment to maintain stability and purity.

Specification

Item	Specification
Appearance	White to off-white powder
Identification (HPLC)	Conforms
Identification (IR)	Conforms to reference spectrum
Assay (HPLC)	≥98.0%
Water Content (KF)	≤1.0%
Residue on Ignition	≤0.1%
Heavy Metals	≤20 ppm
Related Substances (HPLC)	Total impurities ≤2.0%

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.