Description

4-((4-Methylpiperazin-1-Yl)Methyl)Phenylboronic Acid is a high-value boronic acid derivative featuring a piperazine moiety, making it a versatile and critical building block in modern synthetic chemistry. Its primary value lies in its role as a key intermediate in the synthesis of complex pharmaceutical compounds, particularly through Suzuki-Miyaura cross-coupling reactions. This compound is essential for research and development chemists and manufacturers in the pharmaceutical, agrochemical, and advanced materials sectors who require reliable, high-purity intermediates for constructing novel molecular architectures.

Application

• Pharmaceutical Intermediate: A crucial building block in the synthesis of active pharmaceutical ingredients (APIs), especially for kinase inhibitors and other targeted therapies.
• Suzuki-Miyaura Cross-Coupling Reagent: Used extensively in palladium-catalyzed reactions to form carbon-carbon bonds, enabling the construction of complex biaryl structures common in drug discovery.
• Agrochemical Research: Serves as an intermediate in the development of novel herbicides, fungicides, and plant growth regulators.
• Material Science: Employed in the synthesis of organic electronic materials, such as those used in OLEDs and organic semiconductors.
• Chemical Biology & Proteomics: Utilized in the development of molecular probes and affinity ligands for studying biological systems.
• Custom Synthesis & Contract Manufacturing: A key starting material for custom synthesis houses serving the life sciences industry.

Basic Information

Item	Details
Product Name	4-((4-Methylpiperazin-1-Yl)Methyl)Phenylboronic Acid
CAS No.	763120-62-3
Molecular Formula	C13H21BN2O2
Molecular Weight	248.13 g/mol
Synonyms	[4-(4-Methyl-1-piperazinylmethyl)phenyl]boronic acid; 4-(4-Methylpiperazin-1-ylmethyl)benzeneboronic acid; 4-(4-Methylpiperazine-1-ylmethyl)phenylboronic acid; (4-((4-Methylpiperazin-1-yl)methyl)phenyl)boronic acid; B-[4-[(4-Methyl-1-piperazinyl)methyl]phenyl]boronic acid; 763120-62-3; Boronic acid, B-[4-[(4-methyl-1-piperazinyl)methyl]phenyl]-; 4-(N-Methylpiperazinomethyl)phenylboronic acid
EINECS	Contact for details

Quality Control

Our 4-((4-Methylpiperazin-1-Yl)Methyl)Phenylboronic Acid is manufactured under strict quality management systems. Each batch undergoes rigorous analytical testing, including HPLC, NMR, and elemental analysis, to ensure high purity and consistent performance in sensitive applications like pharmaceutical synthesis. Certificates of Analysis (COA) detailing batch-specific results are available upon request, supporting your quality assurance and regulatory documentation needs.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry, and well-ventilated area at a controlled room temperature (15-25°C). Due to its hygroscopic (moisture-sensitive) nature, the container must be kept sealed under an inert atmosphere (e.g., nitrogen or argon) after opening to prevent degradation.

Specification

Item	Specification
Appearance	White to off-white powder
Identification (IR)	Conforms to structure
Purity (HPLC)	≥ 97.0%
Water Content (KF)	≤ 1.0%
Heavy Metals	≤ 20 ppm
Residue on Ignition	≤ 0.1%

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.