Description

4-(2-Methoxyethylamino)Piperidine-1-Carboxylic Acid tert-Butyl Ester is a high-purity, advanced pharmaceutical intermediate of significant commercial importance. This compound is valued for its role as a critical building block in the synthesis of complex active pharmaceutical ingredients (APIs), particularly in central nervous system (CNS) and other therapeutic areas. It is primarily sought by research institutions, contract development and manufacturing organizations (CDMOs), and pharmaceutical companies engaged in innovative drug development and process chemistry.

Application

• Pharmaceutical Intermediate: A key synthetic precursor in the development of novel drug candidates, particularly those targeting neurological and psychiatric disorders.
• API Synthesis: Used as a versatile building block for constructing complex molecular scaffolds in the final stages of Active Pharmaceutical Ingredient (API) manufacturing.
• Medicinal Chemistry Research: Essential for structure-activity relationship (SAR) studies and lead optimization in early-stage drug discovery programs.
• Process Chemistry & Scale-Up: Employed in the development and optimization of scalable, cost-effective synthetic routes for commercial pharmaceutical production.
• Custom Synthesis: Serves as a starting material for the custom synthesis of specialized derivatives and analogs for proprietary research.

Basic Information

Product Name	4-(2-Methoxyethylamino)Piperidine-1-Carboxylic Acid tert-Butyl Ester
CAS No.	710972-40-0
Molecular Formula	C13H26N2O3
Molecular Weight	258.36 g/mol
Synonyms	1-Boc-4-(2-Methoxyethylamino)piperidine; tert-Butyl 4-[(2-methoxyethyl)amino]piperidine-1-carboxylate; 4-[(2-Methoxyethyl)amino]-1-piperidinecarboxylic Acid 1,1-Dimethylethyl Ester; 1,1-Dimethylethyl 4-[(2-Methoxyethyl)amino]-1-piperidinecarboxylate; N-Boc-4-(2-Methoxyethylamino)piperidine; 4-(2-Methoxyethylamino)-1-Boc-piperidine; 1-Boc-4-(2-Methoxyethylamino)piperidine; 4-(2-Methoxyethylamino)piperidine-1-carboxylic acid tert-butyl ester
EINECS	Contact for details

Quality Control

Our production of 4-(2-Methoxyethylamino)Piperidine-1-Carboxylic Acid tert-Butyl Ester adheres to stringent quality management protocols to ensure batch-to-batch consistency and high purity. Each lot is subjected to comprehensive analytical testing, including HPLC, GC, NMR, and mass spectrometry, to confirm identity, purity, and impurity profiles. A detailed Certificate of Analysis (COA) is provided with every shipment, documenting full compliance with agreed specifications. Our quality systems are designed to support cGMP and ICH guidelines for pharmaceutical intermediates.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry, and well-ventilated place at a controlled room temperature (typically 15-25°C). Due to its hygroscopic nature, the container must be kept tightly sealed to prevent moisture absorption, which may affect product stability and performance. For long-term storage, consider using desiccants or storing under an inert atmosphere.

Specification

Item	Specification
Appearance	White to off-white solid
Identification (IR)	Conforms to structure
Identification (NMR)	Conforms to structure
Purity (HPLC)	≥ 98.0%
Water Content (KF)	≤ 0.5%
Residue on Ignition	≤ 0.1%
Heavy Metals	≤ 10 ppm

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.