Description

Cinolazepam CAS NO 75696-02-5 is a high-purity benzodiazepine derivative, recognized for its specific pharmacological profile. This compound is of significant interest for research and development within the pharmaceutical and life sciences sectors. It serves as a critical intermediate and reference standard for scientists and manufacturers developing novel therapeutic agents and analytical methods.

Application

• Pharmaceutical Research & Development: As a key intermediate in the synthesis of novel benzodiazepine-based active pharmaceutical ingredients (APIs).
• Reference Standard: Used in analytical laboratories for method development, validation, and quality control testing via HPLC, GC, or LC-MS.
• Biochemical Studies: Employed in preclinical research to investigate the structure-activity relationships (SAR) of benzodiazepines and their interaction with GABA-A receptors.
• Contract Manufacturing: Supplied to CDMOs (Contract Development and Manufacturing Organizations) for custom synthesis projects and scale-up production.
• Academic Research: Utilized in university and institutional labs for pharmacological and neurochemical studies.

Basic Information

Product Name	Cinolazepam
CAS No.	75696-02-5
Molecular Formula	C₁₈H₁₇ClN₂O₂
Molecular Weight	328.79 g/mol
Synonyms	Cinolazepam; 7-Chloro-5-(2-fluorophenyl)-1,3-dihydro-3-hydroxy-1-(2-propynyl)-2H-1,4-benzodiazepin-2-one; 3-Hydroxyprazepam; 3-OH-Prazepam; 7-Chloro-1-(2-propynyl)-5-(o-fluorophenyl)-1,3-dihydro-3-hydroxy-2H-1,4-benzodiazepin-2-one; Gerodorm; (3S)-7-Chloro-5-(2-fluorophenyl)-1-(prop-2-yn-1-yl)-1,3-dihydro-3-hydroxy-2H-1,4-benzodiazepin-2-one
EINECS	Contact for details

Quality Control

Our Cinolazepam is manufactured under strict quality management systems. Each batch undergoes comprehensive analytical testing to ensure identity, purity, and consistency, meeting the stringent requirements for research and pharmaceutical intermediate applications. A detailed Certificate of Analysis (COA) is provided with every shipment, confirming compliance with agreed specifications.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry, and well-ventilated area at controlled room temperature (typically 15-25°C). Keep away from incompatible materials.

Specification

Item	Specification
Appearance	White to off-white crystalline powder
Identification (IR)	Conforms to reference spectrum
Identification (HPLC)	Retention time matches reference standard
Assay (HPLC)	≥98.0%
Related Substances (HPLC)	Total impurities ≤2.0%
Loss on Drying	≤0.5%
Residue on Ignition	≤0.1%

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.