Description

4-[[(5,7-Diaminopyrido[3,4-B]Pyrazin-3-Yl)Methyl]Amino]Benzoic Acid is a high-purity, advanced pharmaceutical intermediate characterized by its complex heterocyclic structure. This compound is of significant value for its role as a key building block in the synthesis of novel, targeted therapeutic agents. It is primarily sought after by research institutions and pharmaceutical companies engaged in the development of small molecule drugs, particularly in oncology and other specialized therapeutic areas. The CAS number for this compound is 74023-42-0.

Application

This specialized intermediate serves critical functions in advanced chemical synthesis and research. Its primary applications include:

• Pharmaceutical Intermediate: A crucial precursor in the multi-step synthesis of complex active pharmaceutical ingredients (APIs) for investigational new drugs.
• Oncology Drug Research: Serves as a core scaffold for developing novel kinase inhibitors and other targeted cancer therapies.
• Chemical Biology & Proteomics: Used in the design and synthesis of molecular probes for studying enzyme function and protein-protein interactions.
• Academic & Contract Research: Employed in university and CRO laboratories for medicinal chemistry programs and structure-activity relationship (SAR) studies.
• High-Value Fine Chemical Synthesis: Integral to the production of other sophisticated fine chemicals and advanced intermediates with specific biological activity.

Basic Information

Product Name	4-[[(5,7-Diaminopyrido[3,4-B]Pyrazin-3-Yl)Methyl]Amino]Benzoic Acid
CAS No.	74023-42-0
Molecular Formula	C₁₅H₁₅N₇O₂
Molecular Weight	325.33 g/mol
Synonyms	4-{[(5,7-Diaminopyrido[3,4-b]pyrazin-3-yl)methyl]amino}benzoic acid; Benzoic acid, 4-[[(5,7-diaminopyrido[3,4-b]pyrazin-3-yl)methyl]amino]-; 74023-42-0; 5,7-Diamino-3-[(4-carboxyphenylamino)methyl]pyrido[3,4-b]pyrazine
EINECS	Contact for details

Quality Control

We supply this intermediate under strict quality protocols to ensure batch-to-batch consistency for critical research and development. Our products undergo rigorous quality testing, including advanced chromatographic methods, to ensure compliance with client specifications. A comprehensive Certificate of Analysis (COA) detailing purity, identity, and impurity profiles is provided with each batch. We support development under cGMP guidelines where required for pre-clinical and clinical stage manufacturing.

Storage

Preserve in a tightly closed container, protected from light. Due to its hygroscopic (moisture-sensitive) nature, store under dry, inert conditions at a controlled room temperature (15-25°C). For long-term stability, consider storage in a desiccator or under a nitrogen atmosphere.

Specification

Item	Specification
Appearance	Yellow to brown powder
Identification (IR)	Conforms to structure
Purity (HPLC)	≥ 97.0%
Loss on Drying	≤ 2.0%
Residue on Ignition	≤ 0.5%
Heavy Metals	≤ 20 ppm

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.