Description

Tasimelteon CAS NO 609799-22-6 is a selective agonist for the melatonin MT1 and MT2 receptors, developed for the treatment of circadian rhythm sleep disorders. This compound is of significant interest in the pharmaceutical industry for its targeted mechanism of action in regulating the sleep-wake cycle. It is primarily required by pharmaceutical manufacturers and research institutions engaged in the development and production of advanced therapeutics for non-24-hour sleep-wake disorder and other circadian rhythm abnormalities.

Application

• Active Pharmaceutical Ingredient (API) for the manufacture of prescription sleep medications.
• Reference Standard in analytical laboratories for quality control and method validation.
• Biochemical Research for studying melatonin receptor signaling pathways and circadian biology.
• Pharmaceutical Development in pre-formulation studies and dosage form design.
• Clinical Research Material for investigational new drug (IND) applications and trials.

Basic Information

Product Name	Tasimelteon
CAS No.	609799-22-6
Molecular Formula	C₁₅H₁₀N₂O₂
Molecular Weight	250.26 g/mol
Synonyms	VEC-162; BMS-214,778; (1R-trans)-N-[[2-(2,3-Dihydro-1-benzofuran-4-yl)cyclopropyl]methyl]propanamide; Hetlioz (Brand Name); Circadin (related therapeutic area); MT1/MT2 Receptor Agonist
EINECS	Contact for details

Quality Control

Our Tasimelteon is manufactured under strict quality management systems. Each batch undergoes comprehensive analytical testing to ensure it meets high-purity standards suitable for pharmaceutical applications. Certificates of Analysis (COA) are provided, detailing parameters such as assay, related substances, and residual solvents. We adhere to cGMP guidelines where applicable to support our clients' regulatory requirements.

Storage

Preserve in a tightly closed container, protected from light. Store at controlled room temperature, 15-25°C (59-77°F). Keep the container in a dry, well-ventilated area. For long-term storage, consider conditions under an inert atmosphere to ensure stability.

Specification

Item	Specification
Appearance	White to off-white powder
Identification (IR)	Conforms to reference spectrum
Identification (HPLC)	Retention time matches reference standard
Assay (HPLC)	≥ 98.5%
Related Substances (HPLC)	Total impurities ≤ 1.0% Any single impurity ≤ 0.5%
Residual Solvents (GC)	Complies with ICH Q3C guidelines
Loss on Drying	≤ 0.5%
Heavy Metals	≤ 20 ppm

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.