Description

5-Bromo-3-Methyl-2-(Morpholino)Pyridine is a high-purity, advanced pharmaceutical intermediate characterized by its unique pyridine core substituted with bromine, methyl, and morpholino functional groups. This compound is critical for medicinal chemistry research and development, serving as a versatile building block for the synthesis of novel active pharmaceutical ingredients (APIs). It is primarily utilized by R&D chemists and process development scientists in the pharmaceutical, agrochemical, and specialty chemical industries seeking to develop new therapeutic agents and functional materials.

Application

• Pharmaceutical Intermediate: A key precursor in the synthesis of complex drug candidates, particularly those targeting kinase inhibition and central nervous system (CNS) disorders.
• Medicinal Chemistry Research: Used extensively in hit-to-lead and lead optimization campaigns to explore structure-activity relationships (SAR) and improve pharmacokinetic properties.
• Agrochemical Development: Serves as a building block for creating novel pesticides and herbicides with specific modes of action.
• Chemical Biology Probes: Employed in the design and synthesis of molecular probes for studying biological pathways and target validation.
• Ligand Synthesis: Useful for constructing sophisticated ligands in catalysis and material science applications.
• Custom Synthesis & Contract Manufacturing: Supplied to CDMOs (Contract Development and Manufacturing Organizations) for custom synthesis projects under cGMP or research-grade conditions.

Basic Information

Product Name	5-Bromo-3-Methyl-2-(Morpholino)Pyridine
CAS No.	566158-47-2
Molecular Formula	C11H15BrN2O
Molecular Weight	271.16 g/mol
Synonyms	2-(4-Morpholinyl)-5-bromo-3-methylpyridine; 5-Bromo-3-methyl-2-morpholinopyridine; 5-Bromo-3-methyl-2-(4-morpholinyl)pyridine; 2-Morpholino-5-bromo-3-methylpyridine; Pyridine, 5-bromo-3-methyl-2-(4-morpholinyl)-; 566158-47-2
EINECS	Contact for details

Quality Control

Our 5-Bromo-3-Methyl-2-(Morpholino)Pyridine is manufactured under strict quality management systems. Every batch undergoes rigorous analytical testing, including HPLC for purity and NMR/IR for structural confirmation, to ensure it meets the high standards required for research and development. Certificates of Analysis (COA) with detailed chromatographic data are provided for full traceability and quality assurance.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry, and well-ventilated place at room temperature (15-25°C). Keep the container tightly sealed to protect from moisture.

Specification

Item	Specification
Appearance	White to off-white crystalline powder
Identification (IR)	Conforms to structure
Identification (HPLC)	Retention time matches reference standard
Purity (HPLC)	≥ 98.0%
Water Content (KF)	≤ 0.5%
Residue on Ignition	≤ 0.1%

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.