Description

cis-tert-Butyl 3,4-Diazidopyrrolidine-1-Carboxylate is a high-value, multifunctional organic building block characterized by its unique pyrrolidine scaffold bearing two azide groups and a tert-butoxycarbonyl (Boc) protecting group. This compound is essential for advanced organic synthesis, particularly in click chemistry and the construction of complex nitrogen-containing heterocycles. It is primarily utilized by research and development chemists in the pharmaceutical, agrochemical, and materials science industries for the development of novel active ingredients and functional polymers.

Application

• Pharmaceutical Intermediate: A key precursor in the synthesis of novel drug candidates, particularly those targeting neurological disorders and infectious diseases.
• Click Chemistry Reagent: The dual azide functionality enables efficient Huisgen 1,3-dipolar cycloaddition reactions with alkynes to form triazole linkages, a cornerstone of bioconjugation and polymer chemistry.
• Agrochemical Synthesis: Used in the research and development of new herbicides and insecticides with enhanced efficacy and selectivity.
• Polymer & Material Science: Serves as a monomer or cross-linking agent for creating advanced polymers with specific thermal or mechanical properties.
• Chemical Biology Probe Development: Facilitates the labeling and study of biomolecules in proteomics and genomics research.
• Ligand & Catalyst Development: The structured pyrrolidine core is valuable for constructing chiral ligands and organocatalysts used in asymmetric synthesis.

Basic Information

Product Name	cis-tert-Butyl 3,4-Diazidopyrrolidine-1-Carboxylate
CAS No.	480450-25-7
Molecular Formula	C9H15N5O2
Molecular Weight	225.25 g/mol
Synonyms	1-Boc-3,4-diazidopyrrolidine; tert-Butyl 3,4-diazidopyrrolidine-1-carboxylate; 3,4-Diazido-1-(tert-butoxycarbonyl)pyrrolidine; 1-N-Boc-3,4-diazidopyrrolidine; Pyrrolidine-1-carboxylic acid, 3,4-diazido-, 1,1-dimethylethyl ester; (3R,4R)-tert-Butyl 3,4-diazidopyrrolidine-1-carboxylate (for specific stereoisomer); BOC-DAP
EINECS	Contact for details

Quality Control

Every batch of cis-tert-Butyl 3,4-Diazidopyrrolidine-1-Carboxylate is manufactured under strict quality management systems. Our products undergo rigorous analytical testing, including HPLC, NMR, and IR spectroscopy, to ensure high purity and consistent chemical identity. A comprehensive Certificate of Analysis (COA) detailing purity, assay, and impurity profiles is provided with each shipment to support your quality assurance and regulatory documentation needs.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry, and well-ventilated place at a controlled room temperature (15-25°C). This compound is light-sensitive and should be handled under an inert atmosphere when appropriate for prolonged procedures. Keep away from heat, sparks, open flames, and strong oxidizing agents.

Specification

Item	Specification
Appearance	Colorless to pale yellow liquid or low-melting solid
Identification (IR)	Conforms to structure
Purity (HPLC)	≥ 95%
Water Content (KF)	≤ 0.5%
Residual Solvents (GC)	Meets ICH guidelines

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.