Description

2-Azido-1-Methylbenzimidazole is a specialized heterocyclic organic compound featuring an azido functional group, making it a valuable intermediate for click chemistry and other synthetic transformations. Its primary commercial value lies in its role as a versatile building block for the development of pharmaceuticals, agrochemicals, and advanced materials. This product is essential for research and development chemists in the pharmaceutical, biotechnology, and fine chemical industries seeking to incorporate the benzimidazole scaffold into novel molecular entities.

Application

• Pharmaceutical Intermediate: A key precursor in the synthesis of novel drug candidates, particularly those targeting various enzyme systems where the benzimidazole core is pharmacologically active.
• Agrochemical Synthesis: Used in the development of new fungicides, herbicides, and insecticides that leverage the biological activity of azido and benzimidazole components.
• Click Chemistry Reagent: Serves as a critical azide component in copper-catalyzed azide-alkyne cycloaddition (CuAAC) reactions for bioconjugation, polymer chemistry, and material surface functionalization.
• Polymer & Material Science: Employed in the creation of functional polymers, cross-linking agents, and smart materials that require specific chemical reactivity.
• Research & Development: A valuable tool for academic and industrial R&D laboratories exploring new synthetic pathways and heterocyclic chemistry.
• Ligand & Catalyst Development: Used in the preparation of novel ligands and organocatalysts for asymmetric synthesis and metal complexation.

Basic Information

Product Name	2-Azido-1-Methylbenzimidazole
CAS No.	1516-73-0
Molecular Formula	C8H7N5
Molecular Weight	173.17 g/mol
Synonyms	1-Methyl-2-azidobenzimidazole; 2-Azido-1-methyl-1H-benzimidazole; 1-Methyl-2-azido-1H-benzimidazole; 2-Azido-1-methylbenzimidazole; 1516-73-0; Azidomethylbenzimidazole; NSC 406021; 1H-Benzimidazole, 2-azido-1-methyl-
EINECS	Contact for details

Quality Control

Our 2-Azido-1-Methylbenzimidazole is manufactured under strict quality management systems to ensure batch-to-batch consistency and high purity. Each lot undergoes comprehensive analytical testing, including HPLC for assay and purity, and is supplied with a detailed Certificate of Analysis (COA). We are committed to meeting the stringent requirements of our global customers in research and cGMP environments.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry, well-ventilated place at a controlled room temperature (15-25°C). Due to its nature as an azide compound and being easily oxidized, it is recommended to store under an inert atmosphere (e.g., nitrogen or argon) for long-term stability. Keep away from heat, sparks, open flames, and incompatible materials.

Specification

Item	Specification
Appearance	Off-white to light yellow crystalline powder
Identification (IR)	Conforms to structure
Assay (HPLC)	≥ 97.0%
Purity (HPLC)	≥ 98.0%
Melting Point	Contact for details
Loss on Drying	≤ 0.5%
Residue on Ignition	≤ 0.1%
Heavy Metals	≤ 20 ppm

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.