Description

4-(5-Iodo-Pyridin-2-Yl)-Morpholine is a high-purity, advanced pharmaceutical intermediate featuring a substituted pyridine core with a morpholine moiety. This compound is critical for medicinal chemistry research and development, serving as a versatile building block for the synthesis of novel active pharmaceutical ingredients (APIs). It is primarily utilized by R&D chemists and process development scientists in the pharmaceutical, agrochemical, and specialty chemical industries seeking to develop new drug candidates and fine chemicals.

Application

• Pharmaceutical Intermediate: A key precursor in the synthesis of complex molecules for drug discovery programs, particularly in oncology and CNS therapeutic areas.
• Medicinal Chemistry Building Block: Used for structure-activity relationship (SAR) studies and lead optimization due to its halogenated heterocyclic structure.
• Agrochemical Research: Serves as a synthetic intermediate in the development of new crop protection agents and pesticides.
• Ligand Synthesis: Employed in the preparation of specialized ligands for catalysis and material science applications.
• Chemical Biology Probes: Utilized in the design and synthesis of molecular probes for studying biological pathways and target engagement.

Basic Information

Product Name	4-(5-Iodo-Pyridin-2-Yl)-Morpholine
CAS No.	470463-42-4
Molecular Formula	C9H11IN2O
Molecular Weight	290.10 g/mol
Synonyms	4-(5-Iodopyridin-2-yl)morpholine; 2-Morpholino-5-iodopyridine; 5-Iodo-2-morpholinopyridine; Morpholine, 4-(5-iodo-2-pyridinyl)-; 470463-42-4; 4-(5-Iodo-2-pyridinyl)morpholine
EINECS	Contact for details

Quality Control

Our 4-(5-Iodo-Pyridin-2-Yl)-Morpholine is manufactured under strict quality management systems. Each batch undergoes comprehensive analytical testing, including HPLC, NMR, and mass spectrometry, to ensure identity, purity, and consistency. We provide full traceability and Certificates of Analysis (COA) are available for all shipments, confirming compliance with customer specifications and internal quality standards.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry, well-ventilated area at controlled room temperature (15-25°C). Keep away from incompatible materials. The product is light-sensitive and should be handled accordingly to maintain stability.

Specification

Item	Specification
Appearance	White to off-white crystalline powder
Identification (IR)	Conforms to structure
Identification (NMR)	Conforms to structure
Purity (HPLC)	≥ 97.0%
Water Content (KF)	≤ 0.5%
Residue on Ignition	≤ 0.1%

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.