Description

4-(3-Iodo-Pyridin-2-Yl)-Morpholine is a high-value, heterocyclic organic building block featuring a pyridine core substituted with iodine and a morpholine ring. This compound is critical for medicinal chemistry research and pharmaceutical development, serving as a versatile intermediate for constructing complex molecules. It is primarily sought after by R&D chemists and process development scientists in the pharmaceutical, agrochemical, and advanced material sectors for applications in drug discovery and synthesis.

Application

• Pharmaceutical Intermediate: Key building block for the synthesis of potential active pharmaceutical ingredients (APIs), particularly in kinase inhibitor and central nervous system (CNS) drug discovery programs.
• Medicinal Chemistry Research: Used in structure-activity relationship (SAR) studies and lead optimization due to its modifiable iodine handle for cross-coupling reactions.
• Agrochemical Synthesis: Intermediate in the development of novel crop protection agents and herbicides.
• Chemical Biology Probes: Utilized in the creation of molecular probes for studying biological pathways and target engagement.
• Material Science: Potential precursor for the synthesis of specialized ligands in catalysis or functional organic materials.
• Contract Research & Manufacturing (CRO/CMO): Supplied to organizations offering custom synthesis and process development services.

Basic Information

Product Name	4-(3-Iodo-Pyridin-2-Yl)-Morpholine
CAS No.	470463-40-2
Molecular Formula	C9H11IN2O
Molecular Weight	290.10 g/mol
Synonyms	4-(3-Iodopyridin-2-yl)morpholine; 2-Morpholino-3-iodopyridine; 3-Iodo-2-(4-morpholinyl)pyridine; 3-Iodo-2-morpholinopyridine; 470463-40-2; 4-(3-Iodo-2-pyridinyl)morpholine; 4-(3-Iodopyridin-2-yl)-morpholine; 4-(3-Iodo-2-pyridyl)morpholine
EINECS	Contact for details

Quality Control

Our 4-(3-Iodo-Pyridin-2-Yl)-Morpholine is manufactured under strict quality management systems. Each batch undergoes rigorous analytical testing to ensure high purity and consistency, meeting the stringent requirements for research and development use. A comprehensive Certificate of Analysis (COA) detailing purity, identity, and impurity profiles is provided with every shipment to guarantee traceability and compliance with your specifications.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry, and well-ventilated place at room temperature (15-25°C). Keep away from incompatible materials. Due to its light-sensitive nature, prolonged exposure to light should be avoided.

Specification

Item	Specification
Appearance	White to off-white crystalline powder
Identification (IR)	Conforms to structure
Purity (HPLC)	≥ 97.0%
Water Content (KF)	≤ 0.5%
Residue on Ignition	≤ 0.1%

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.