Description

1,2-Diazaspiro[2.5]Oct-1-Ene-6-Carboxylic Acid is a high-value, spirocyclic heterocyclic compound featuring a fused diaziridine and carboxylic acid functionality. This unique structure makes it a critical advanced pharmaceutical intermediate and a versatile building block in organic synthesis. It is primarily utilized by R&D chemists and process development scientists in the pharmaceutical, agrochemical, and specialty chemical industries for constructing complex molecular architectures.

Application

• Pharmaceutical Intermediate: A key precursor in the synthesis of novel active pharmaceutical ingredients (APIs), particularly those targeting central nervous system (CNS) disorders and metabolic diseases.
• Agrochemical Research: Serves as a building block for developing new herbicides, fungicides, and insecticides with novel modes of action.
• Chemical Biology Probe: Used in medicinal chemistry for structure-activity relationship (SAR) studies and as a scaffold for designing enzyme inhibitors or receptor modulators.
• Material Science: Potential monomer or cross-linking agent for creating polymers with specific thermal or mechanical properties.
• Academic & Contract Research: Employed in university and CRO laboratories for methodological development and exploring new chemical spaces in heterocyclic chemistry.

Basic Information

Product Name	1,2-Diazaspiro[2.5]Oct-1-Ene-6-Carboxylic Acid
CAS No.	36908-76-6
Molecular Formula	C7H10N2O2
Molecular Weight	154.17 g/mol
Synonyms	6-Carboxy-1,2-diazaspiro[2.5]oct-1-ene; 1,2-Diazaspiro[2.5]oct-1-ene-6-carboxylic acid; Diazaspirooctenecarboxylic acid; Spiro[diaziridine-3,1'-cyclopentane]-2-carboxylic acid; 1-Azaspiro[2.5]oct-1-ene-2-carboxylic acid (related structure); CAS 36908-76-6
EINECS	Contact for details

Quality Control

Our production of 1,2-Diazaspiro[2.5]Oct-1-Ene-6-Carboxylic Acid adheres to stringent in-process controls and final release testing. Each batch is analyzed to ensure high chemical purity and structural integrity, with specifications tailored to research and GMP-grade requirements. Comprehensive Certificates of Analysis (COA) detailing identity, purity (HPLC), and impurity profiles are provided with every shipment.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry place at a controlled room temperature (15-25°C). This compound is hygroscopic (moisture-sensitive); therefore, the container must be kept tightly sealed in a dry environment to prevent degradation. For long-term storage, consider using desiccants.

Specification

Item	Specification
Appearance	White to off-white crystalline powder
Identification (IR)	Conforms to structure
Purity (HPLC)	≥ 97.0%
Water Content (KF)	≤ 1.0%
Residue on Ignition	≤ 0.1%
Single Unknown Impurity (HPLC)	≤ 1.0%
Total Impurities (HPLC)	≤ 3.0%

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.