Description

(3S,4S)-3,4-Diazido-1-(Phenylmethyl)Pyrrolidine is a high-value, stereochemically defined organic building block featuring a diazido-functionalized pyrrolidine core. This compound is of significant interest in advanced organic synthesis, particularly for applications requiring precise spatial orientation and click chemistry reactivity. It serves as a critical intermediate for researchers and manufacturers in the pharmaceutical and agrochemical sectors, enabling the development of novel active ingredients and complex molecular architectures.

Application

• Pharmaceutical Intermediate: A key chiral synthon for the synthesis of potential drug candidates, including protease inhibitors and other biologically active molecules.
• Click Chemistry Reagent: Utilized in copper-catalyzed azide-alkyne cycloaddition (CuAAC) reactions to efficiently construct complex heterocyclic systems or conjugate molecules.
• Agrochemical Research: Serves as a building block for developing novel pesticides and herbicides with specific stereochemical requirements.
• Material Science: Used in the synthesis of functional polymers and dendrimers where the azide groups facilitate cross-linking or attachment of other functional units.
• Chemical Biology Probes: Enables the labeling and study of biomolecules through bioorthogonal conjugation strategies.
• Academic & R&D: A valuable tool for methodological development in organic synthesis and catalysis studies.

Basic Information

Product Name	(3S,4S)-3,4-Diazido-1-(Phenylmethyl)Pyrrolidine
CAS No.	288313-99-5
Molecular Formula	C11H13N7
Molecular Weight	243.27 g/mol
Synonyms	(3S,4S)-3,4-Diazido-1-benzylpyrrolidine; 1-Benzyl-3,4-diazidopyrrolidine, (3S,4S)-; (3S,4S)-1-Benzyl-3,4-diazidopyrrolidine; (3S,4S)-1-(Phenylmethyl)-3,4-diazidopyrrolidine; 3,4-Diazido-1-benzylpyrrolidine (stereoisomer); Pyrrolidine, 3,4-diazido-1-(phenylmethyl)-, (3S,4S)-; Chiral diazido pyrrolidine; Benzyl-protected diazidopyrrolidine
EINECS	Contact for details

Quality Control

Our (3S,4S)-3,4-Diazido-1-(Phenylmethyl)Pyrrolidine is manufactured under strict quality management systems. Each batch undergoes rigorous analytical testing, including chiral purity verification, to ensure it meets the high standards required for research and process chemistry. Certificates of Analysis (COA) detailing specifications such as enantiomeric excess, chemical purity, and identity confirmation are provided with every shipment.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry, and well-ventilated place, preferably at 2-8°C for long-term stability. This compound is light-sensitive (store away from light) and should be handled with appropriate safety precautions due to the presence of azide functional groups.

Specification

Item	Specification
Appearance	Colorless to pale yellow liquid or low-melting solid
Identification (IR)	Conforms to structure
Purity (HPLC)	≥ 95.0%
Enantiomeric Excess (Chiral HPLC)	≥ 98.0%
Water Content (KF)	≤ 0.5%
Residual Solvents (GC)	Meets ICH guidelines

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.