Description

2,5-Dimethoxypyridine-4-Boronic Acid is a versatile and high-value boronic acid derivative, serving as a critical building block in modern synthetic chemistry. Its primary value lies in its role as a key coupling partner in Suzuki-Miyaura cross-coupling reactions, enabling the efficient construction of complex biaryl and heterobiaryl structures. This compound is essential for researchers and manufacturers in the pharmaceutical, agrochemical, and advanced materials sectors who are developing new active ingredients and functional molecules.

Application

• Pharmaceutical Intermediate: A crucial precursor in the synthesis of active pharmaceutical ingredients (APIs), particularly for drugs targeting the central nervous system, oncology, and inflammation.
• Agrochemical Synthesis: Used to construct novel pyridine-based herbicides, fungicides, and insecticides with improved efficacy and environmental profiles.
• Ligand & Catalyst Development: Serves as a building block for creating sophisticated ligands and organocatalysts used in asymmetric synthesis and other catalytic processes.
• Material Science Research: Employed in the development of organic electronic materials, such as organic light-emitting diodes (OLEDs) and semiconductors, due to its electron-donating methoxy groups.
• Chemical Biology & Probe Synthesis: Utilized for labeling and modifying biomolecules or creating molecular probes for diagnostic and research applications.
• Custom Synthesis & Contract Manufacturing: A key starting material for custom synthesis houses and CDMOs (Contract Development and Manufacturing Organizations) serving global clients.

Basic Information

Product Name	2,5-Dimethoxypyridine-4-Boronic Acid
CAS No.	1630193-77-9
Molecular Formula	C7H10BNO4
Molecular Weight	182.97 g/mol
Synonyms	(2,5-Dimethoxypyridin-4-yl)boronic Acid; 4-Borono-2,5-dimethoxypyridine; 2,5-Dimethoxy-4-pyridineboronic Acid; 4-Pyridineboronic Acid, 2,5-dimethoxy-; 1630193-77-9; 2,5-Dimethoxy-4-pyridinylboronic Acid
EINECS	Contact for details

Quality Control

Every batch of 2,5-Dimethoxypyridine-4-Boronic Acid is produced and tested under strict quality management protocols to ensure consistency and reliability for your critical synthesis. We provide comprehensive Certificates of Analysis (COA) with each shipment, detailing key parameters such as purity (by HPLC), boronic acid content, and impurity profiles. Our quality systems are designed to support cGMP (current Good Manufacturing Practice) requirements for advanced pharmaceutical intermediates.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry, and well-ventilated place at room temperature (15-25°C). This compound is hygroscopic (moisture-sensitive) and should be handled under an inert atmosphere (e.g., nitrogen or argon) for long-term storage or after opening to maintain stability and purity.

Specification

Item	Specification
Appearance	White to off-white powder or crystalline solid
Identification (IR)	Conforms to structure
Purity (HPLC)	≥97.0% (Area %)
Water Content (KF)	≤1.0%
Heavy Metals	≤20 ppm
Residue on Ignition	≤0.1%

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.