Description

4-(Boc-Aminomethyl)Pyridine-2-Carboxylate Sodium is a high-purity, protected amino acid derivative widely used as a critical building block in advanced organic synthesis. Its primary value lies in providing a versatile, Boc-protected aminomethylpyridine scaffold that facilitates the controlled construction of complex molecules, particularly in pharmaceutical research. This compound is essential for medicinal chemists and process development scientists in the pharmaceutical, agrochemical, and specialty chemical industries who require reliable, high-quality intermediates for drug discovery and development programs.

Application

• Pharmaceutical Intermediate: A key building block for the synthesis of active pharmaceutical ingredients (APIs), especially those containing pyridine and amino acid motifs.
• Peptidomimetic Research: Used in the design and synthesis of peptide analogs and mimetics for drug discovery targeting various diseases.
• Ligand Synthesis: Serves as a precursor for creating complex ligands used in catalysis and metal-organic frameworks (MOFs).
• Protease Inhibitor Development: A valuable intermediate in the construction of protease inhibitor candidates, a major class of therapeutic agents.
• Chemical Biology Probes: Employed in the synthesis of molecular probes for studying biological processes and target identification.
• Agrochemical Synthesis: Used as an intermediate in the development of novel herbicides, fungicides, and insecticides.

Basic Information

Product Name	4-(Boc-Aminomethyl)Pyridine-2-Carboxylate Sodium
CAS No.	1185292-66-3
Molecular Formula	C13H17N2NaO4
Molecular Weight	288.28 g/mol
Synonyms	Sodium 4-[[(tert-butoxycarbonyl)amino]methyl]pyridine-2-carboxylate; 2-Pyridinecarboxylic acid, 4-[[[(1,1-dimethylethoxy)carbonyl]amino]methyl]-, sodium salt (1:1); 4-(N-Boc-aminomethyl)picolinic acid sodium salt; Boc-Amp-OMe sodium salt (common abbreviation); Sodium 4-(Boc-aminomethyl)picolinate; tert-Butyl N-[(2-carboxylato-4-pyridyl)methyl]carbamate; 4-(Boc-NH-CH2)-2-PyCOONa
EINECS	Contact for details

Quality Control

Our 4-(Boc-Aminomethyl)Pyridine-2-Carboxylate Sodium is manufactured under strict quality management systems to ensure batch-to-batch consistency and high purity suitable for research and development. Each lot is accompanied by a comprehensive Certificate of Analysis (COA) detailing purity, identity, and impurity profiles. We adhere to relevant industry standards and can provide material tailored to specific project requirements, including custom purity grades.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry, and well-ventilated area at a controlled room temperature (15-25°C). This product is hygroscopic (moisture-sensitive) and should be handled under dry conditions to prevent degradation. For long-term storage, consider storing under an inert atmosphere.

Specification

Item	Specification
Appearance	White to off-white powder
Identification (IR)	Conforms to structure
Identification (NMR)	Conforms to structure
Assay (HPLC)	≥97.0%
Water Content (KF)	≤1.0%
Residue on Ignition	≤0.5%
Heavy Metals	≤20 ppm

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.