Description

5-Bromo-4-Azaindole 3-Carboxylic Acid is a high-purity, advanced pharmaceutical intermediate characterized by its unique heterocyclic structure. This compound is critical for medicinal chemistry research and development, particularly in the synthesis of targeted kinase inhibitors and other biologically active molecules. It is primarily sought by pharmaceutical R&D laboratories and fine chemical manufacturers engaged in developing novel therapeutics for oncology and inflammatory diseases.

Application

• Pharmaceutical Intermediate: A key building block in the synthesis of potent and selective kinase inhibitors for targeted cancer therapies.
• Medicinal Chemistry Research: Used in structure-activity relationship (SAR) studies and lead optimization programs to develop new drug candidates.
• Biochemical Tool Compound: Serves as a core scaffold for developing probes to study specific enzyme pathways and biological mechanisms.
• Fine Chemical Synthesis: Employed in multi-step organic syntheses to create complex, nitrogen-containing heterocycles with potential biological activity.
• Contract Research & Development (CRO/CMO): Supplied to organizations specializing in custom synthesis and process development for the pharmaceutical industry.

Basic Information

Product Name	5-Bromo-4-Azaindole 3-Carboxylic Acid
CAS No.	1167056-46-3
Molecular Formula	C8H5BrN2O2
Molecular Weight	241.04 g/mol
Synonyms	5-Bromo-1H-pyrrolo[3,2-b]pyridine-3-carboxylic acid; 5-Bromo-4-azaindole-3-carboxylic acid; 5-Bromo-1H-pyrrolo[3,2-b]pyridine-3-carboxylic acid; 5-Bromo-7-azaindole-3-carboxylic acid; 3-Carboxy-5-bromo-4-azaindole; 1167056-46-3; 5-Bromo-4-aza-indole-3-carboxylic acid
EINECS	Contact for details

Quality Control

Our 5-Bromo-4-Azaindole 3-Carboxylic Acid is manufactured under strict quality management systems. Every batch undergoes comprehensive analytical testing, including HPLC, NMR, and mass spectrometry, to ensure identity, purity, and consistency. We provide a detailed Certificate of Analysis (COA) with each shipment, confirming compliance with customer specifications and industry best practices for advanced pharmaceutical intermediates.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry, well-ventilated area at controlled room temperature (15-25°C). This material is hygroscopic (moisture-sensitive). Keep away from strong oxidizing agents.

Specification

Item	Specification
Appearance	White to off-white powder
Identification (HPLC)	Conforms
Identification (IR)	Conforms
Purity (HPLC)	≥ 97.0%
Water Content (KF)	≤ 1.0%
Residue on Ignition	≤ 0.5%

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.