Description

1-Boc-3-(2-Cbz-Amino-2-Methoxycarbonyl-Vinyl)Piperidine is a sophisticated, high-purity piperidine derivative designed for advanced pharmaceutical research and development. This compound serves as a critical protected intermediate in the synthesis of complex molecules, enabling the construction of novel drug candidates with precise stereochemistry. It is primarily utilized by medicinal chemists and process development scientists in the pharmaceutical and biotechnology industries for the creation of new therapeutic agents.

Application

• Pharmaceutical Intermediate: A key building block in the synthesis of active pharmaceutical ingredients (APIs), particularly for central nervous system (CNS) and oncology targets.
• Medicinal Chemistry Research: Used in lead optimization and structure-activity relationship (SAR) studies to explore new chemical entities.
• Process Chemistry Development: Serves as a starting material or intermediate in the scale-up and optimization of synthetic routes under GMP conditions.
• Peptidomimetic Synthesis: Facilitates the creation of peptide-like compounds with enhanced metabolic stability and bioavailability.
• Custom Synthesis: Employed by contract research and manufacturing organizations (CROs/CMOs) for client-specific projects requiring complex heterocyclic chemistry.

Basic Information

Product Name	1-Boc-3-(2-Cbz-Amino-2-Methoxycarbonyl-Vinyl)Piperidine
CAS No.	1017789-37-5
Molecular Formula	C22H30N2O6
Molecular Weight	418.49 g/mol
Synonyms	1-Boc-3-[(2-{[(Benzyloxy)carbonyl]amino}-2-methoxy-2-oxoethylidene)]piperidine; tert-Butyl 3-[(Z)-2-{[(benzyloxy)carbonyl]amino}-2-methoxy-2-oxoethylidene]piperidine-1-carboxylate; 1-(tert-Butoxycarbonyl)-3-[(Z)-2-(benzyloxycarbonylamino)-2-methoxy-2-oxoethylidene]piperidine; N-Boc-3-(N-Cbz-amino-methoxycarbonyl-vinyl)piperidine; Piperidine, 1-[(1,1-dimethylethoxy)carbonyl]-3-[(2-{[(phenylmethoxy)carbonyl]amino}-2-methoxy-2-oxoethylidene)]-; BOC-Cbz-Amino-Methoxycarbonyl-Vinyl-Piperidine
EINECS	Contact for details

Quality Control

Our 1-Boc-3-(2-Cbz-Amino-2-Methoxycarbonyl-Vinyl)Piperidine is manufactured under strict quality management systems. Each batch undergoes rigorous analytical testing, including HPLC, NMR, and mass spectrometry, to ensure high chemical purity and structural integrity. Certificates of Analysis (COA) with detailed chromatographic data are available for every lot to support your regulatory and research documentation needs.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry place at a controlled room temperature (15-25°C). The compound is moisture-sensitive; keep the container tightly sealed in a dry environment. For long-term storage, consider storing under an inert atmosphere.

Specification

Item	Specification
Appearance	White to off-white solid
Identification (IR)	Conforms to structure
Identification (NMR)	Conforms to structure
Purity (HPLC)	≥ 97.0%
Water Content (KF)	≤ 0.5%
Residue on Ignition	≤ 0.1%

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.