Description

4-Bromo-5-Azaindole is a high-value brominated heterocyclic building block, specifically a halogenated azaindole derivative. This compound is critical for medicinal chemistry research and development, serving as a versatile scaffold for constructing novel pharmacologically active molecules. It is primarily utilized by pharmaceutical R&D teams and fine chemical manufacturers specializing in the synthesis of targeted small molecule libraries and potential drug candidates.

Application

• Pharmaceutical Intermediate: A key precursor in the synthesis of kinase inhibitors and other targeted therapeutic agents.
• Medicinal Chemistry Research: Used as a core scaffold for structure-activity relationship (SAR) studies and high-throughput screening libraries.
• Organic Synthesis Building Block: Enables functionalization and further cross-coupling reactions (e.g., Suzuki, Buchwald-Hartwig) due to the reactive bromine substituent.
• Agrochemical Development: Serves as an intermediate in the research and synthesis of novel crop protection agents.
• Chemical Biology Probes: Utilized in the development of molecular probes for studying biological pathways and target engagement.

Basic Information

Product Name	4-Bromo-5-Azaindole
CAS No.	1000342-68-6
Molecular Formula	C7H5BrN2
Molecular Weight	197.04 g/mol
Synonyms	4-Bromo-1H-pyrrolo[3,2-b]pyridine; 4-Bromo-7-azaindole; 4-Bromo-1H-pyrrolo[3,2-b]pyridine; 1H-Pyrrolo[3,2-b]pyridine, 4-bromo-; 4-Bromo-pyrrolo[3,2-b]pyridine
EINECS	Contact for details

Quality Control

Our 4-Bromo-5-Azaindole is manufactured under strict quality control protocols to ensure batch-to-batch consistency and high purity, suitable for demanding research applications. We provide comprehensive analytical data, including HPLC purity, NMR, and mass spectrometry confirmation. A Certificate of Analysis (COA) is supplied with each batch to guarantee compliance with your specifications.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry, and well-ventilated place at room temperature (15-25°C). Keep away from incompatible materials.

Specification

Item	Specification
Appearance	White to off-white powder
Identification (HPLC/MS)	Conforms
Purity (HPLC)	≥97.0%
Water Content (KF)	≤0.5%
Residue on Ignition	≤0.1%

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.