Description

3-Iodo-4-Methyl-5-Azaindole is a high-purity, advanced pharmaceutical intermediate belonging to the azaindole class of heterocyclic compounds. This specialized chemical is critical for medicinal chemistry research and the development of novel therapeutic agents, particularly in oncology and antiviral drug discovery. It is primarily utilized by R&D scientists and process chemists in pharmaceutical, biotechnology, and fine chemical synthesis sectors.

Application

• Pharmaceutical Intermediate: Serves as a key building block in the synthesis of complex drug candidates, especially kinase inhibitors and other targeted small-molecule therapies.
• Medicinal Chemistry Research: Used in structure-activity relationship (SAR) studies and lead optimization programs due to its versatile azaindole scaffold.
• Organic Synthesis Reagent: Employed in cross-coupling reactions (e.g., Suzuki, Sonogashira) and other metal-catalyzed transformations to introduce functional complexity.
• Biochemical Probe Development: Acts as a core structure for developing chemical probes to study biological pathways and protein functions.
• Agrochemical Research: Potential application in the research and development of new active ingredients for crop protection.

Basic Information

Product Name	3-Iodo-4-Methyl-5-Azaindole
CAS No.	1000342-66-4
Molecular Formula	C8H7IN2
Molecular Weight	258.06 g/mol
Synonyms	4-Methyl-3-iodo-1H-pyrrolo[3,2-c]pyridine; 3-Iodo-4-methyl-1H-pyrrolo[3,2-c]pyridine; 1H-Pyrrolo[3,2-c]pyridine, 3-iodo-4-methyl-; 4-Methyl-3-iodo-7-azaindole
EINECS	Contact for details

Quality Control

Our 3-Iodo-4-Methyl-5-Azaindole is manufactured under strict quality management systems. Each batch undergoes comprehensive analytical testing, including HPLC for purity, NMR and MS for structural confirmation, and residual solvent analysis to ensure it meets the stringent requirements for pharmaceutical R&D. A detailed Certificate of Analysis (COA) is provided with every shipment, guaranteeing traceability, consistency, and compliance with your specifications.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry, and well-ventilated place at a controlled room temperature (15-25°C). Keep the container sealed to protect this light-sensitive material from moisture and atmospheric contamination.

Specification

Item	Specification
Appearance	White to off-white powder
Identification (HPLC)	Conforms
Identification (NMR)	Conforms
Purity (HPLC)	≥ 97.0%
Water Content (KF)	≤ 0.5%
Residual Solvents (GC)	Meets ICH guidelines

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.