Description

Haloperidol 4-Azidobenzoate is a chemically modified derivative of the antipsychotic agent haloperidol, designed for advanced research and development applications. This compound is of significant interest in pharmaceutical chemistry for its utility as a molecular probe and a potential precursor in the synthesis of novel bioactive conjugates. It serves the needs of research institutions, pharmaceutical R&D laboratories, and fine chemical manufacturers focused on neuropharmacology and targeted drug delivery systems.

Application

• As a key intermediate in the research and synthesis of novel haloperidol analogs and prodrugs.
• Utilized as a biochemical probe in neuroscience research to study dopamine receptor interactions and signaling pathways.
• Potential use in the development of photoaffinity labeling agents for target identification studies.
• Employed in academic and industrial research for structure-activity relationship (SAR) studies of antipsychotic agents.
• Serves as a specialized building block in medicinal chemistry for creating targeted molecular conjugates.
• Used in analytical method development as a reference standard for quality control in pharmaceutical manufacturing.

Basic Information

Product Name	Haloperidol 4-Azidobenzoate
CAS No.	117345-85-4
Molecular Formula	C27H26ClFN4O3
Molecular Weight	508.98 g/mol
Synonyms	4-Azidobenzoic Acid Haloperidol Ester; 1-(4-Fluorophenyl)-4-[4-(4-azidobenzoyl)piperidin-1-yl]butan-1-one; Haloperidol 4-Azidobenzoate Ester; Haloperidol Azidobenzoate; 4-Azidobenzoyl Haloperidol; NSC 339539; Butyrophenone Derivative
EINECS	Contact for details

Quality Control

Our Haloperidol 4-Azidobenzoate is manufactured under strict quality management systems. Each batch undergoes comprehensive analytical testing, including HPLC for purity, IR and NMR for structural confirmation, and residual solvent analysis. We provide full traceability and Certificates of Analysis (COA) are available for all shipments, ensuring compliance with research-grade specifications.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry place at controlled room temperature (15-25°C). The product is light-sensitive and should be handled under appropriate conditions to maintain stability.

Specification

Item	Specification
Appearance	White to off-white solid
Identification (IR)	Conforms to structure
Identification (HPLC)	Retention time matches reference standard
Purity (HPLC)	≥ 98.0%
Related Substances (HPLC)	Total impurities ≤ 2.0%
Water Content (KF)	≤ 0.5%
Residual Solvents (GC)	Complies with ICH guidelines

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.