Tinib Antineoplastic Drugs

Tinib Antineoplastic Drugs

Tinib antineoplastic drugs are a major class of targeted cancer therapies that inhibit dysregulated tyrosine kinases or serine/threonine kinases involved in tumor growth, angiogenesis, and metastasis. Represented by imatinib, erlotinib, gefitinib, sunitinib, sorafenib, and numerous next-generation inhibitors, these APIs block oncogenic signaling pathways such as EGFR, VEGFR, PDGFR, BCR-ABL, ALK, and RET. Their precision targeting enables high efficacy with reduced systemic toxicity compared to traditional chemotherapy. Tinib drugs are widely used in leukemia, lung cancer, renal cancer, gastrointestinal stromal tumors, and melanoma. Resistance caused by kinase mutations has led to the development of multi-targeted and mutation-specific inhibitors, making tinibs a cornerstone of precision oncology.

Sar131675 CAS NO 1092538-80-1

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CAS No.:1092538-80-1

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3-(3-Fluoro-5-Methoxyphenyl)-1H-Pyrazolo[3,4-D]Pyrimidin-4-Amine CAS NO 1092789-24-6

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CAS No.:1092789-24-6

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Ruxolitinib Phosphate CAS NO 1092939-17-7

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CAS No.:1092939-17-7

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B-Raf Inhibitor 1 CAS NO 1093100-40-3

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CAS No.:1093100-40-3

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Idx-989 CAS NO 1097733-15-7

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CAS No.:1097733-15-7

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Tepotinib CAS NO 1100598-32-0

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CAS No.:1100598-32-0

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Azd3147 CAS NO 1101810-02-9

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CAS No.:1101810-02-9

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Entrectinib CAS NO 1108743-60-7

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CAS No.:1108743-60-7

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