Description

1-(1-Benzyl-Piperidin-4-Yl)-Azetidine-3-Carboxylic Acid is a high-purity, advanced pharmaceutical intermediate with a complex heterocyclic structure. This compound is critical for the research and development of novel therapeutic agents, particularly in the field of central nervous system (CNS) and metabolic disorder treatments. It is primarily sought by pharmaceutical R&D laboratories, contract research organizations (CROs), and fine chemical manufacturers for use in drug discovery and process chemistry.

Application

• Pharmaceutical Intermediate: A key building block in the synthesis of potent and selective drug candidates targeting G-protein-coupled receptors (GPCRs).
• Medicinal Chemistry Research: Used in structure-activity relationship (SAR) studies and lead optimization programs for new chemical entities.
• Neurological Disorder Drug Development: Serves as a core scaffold for molecules being investigated for conditions such as Alzheimer's disease, schizophrenia, and Parkinson's disease.
• Chemical Biology Probes: Utilized in the development of tool compounds for studying biological pathways and target validation.
• Process Development & Scale-up: Employed in the development of robust and scalable synthetic routes for active pharmaceutical ingredients (APIs).
• Custom Synthesis: A starting material for the custom synthesis of more complex, proprietary molecules for client-specific research programs.

Basic Information

Product Name	1-(1-Benzyl-Piperidin-4-Yl)-Azetidine-3-Carboxylic Acid
CAS No.	889952-36-7
Molecular Formula	C16H22N2O2
Molecular Weight	274.36 g/mol
Synonyms	1-(1-Benzylpiperidin-4-yl)azetidine-3-carboxylic acid; Azetidine-3-carboxylic acid, 1-(1-benzyl-4-piperidinyl)-; 1-(1-Benzyl-piperidin-4-yl)-azetidine-3-carboxylic acid; 1-(1-Benzylpiperidin-4-yl)azetidine-3-carboxylic acid; 889952-36-7; 1-(1-Benzyl-4-piperidyl)azetidine-3-carboxylic acid; 1-(1-Benzylpiperidin-4-yl)azetidine-3-carboxylate
EINECS	Contact for details

Quality Control

Our 1-(1-Benzyl-Piperidin-4-Yl)-Azetidine-3-Carboxylic Acid is manufactured under strict quality management systems. Each batch undergoes comprehensive analytical testing, including HPLC, NMR, and mass spectrometry, to ensure identity, purity, and consistency. We provide a detailed Certificate of Analysis (COA) with every shipment, confirming compliance with customer specifications and current industry standards for advanced pharmaceutical intermediates.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry, and well-ventilated place at a controlled room temperature (15-25°C). This material is hygroscopic (moisture-sensitive); the container must be kept tightly sealed in a dry environment to prevent degradation.

Specification

Item	Specification
Appearance	White to off-white solid
Identification (IR)	Conforms to structure
Identification (NMR)	Conforms to structure
Purity (HPLC)	≥ 97.0%
Water Content (KF)	≤ 1.0%
Residue on Ignition	≤ 0.5%

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.