Description

1-Boc-4-Methyl-4-Morpholin-4-Yl-Piperidine is a high-purity, advanced pharmaceutical intermediate crucial for modern drug discovery and development. This compound serves as a key protected building block for synthesizing complex molecules, particularly in medicinal chemistry programs targeting central nervous system (CNS) disorders. It is primarily utilized by research institutions and pharmaceutical companies engaged in the development of novel therapeutic agents, where its structural features enable precise molecular modifications. The product is supplied with stringent quality control to ensure batch-to-batch consistency for reliable research and scale-up processes.

Application

• Pharmaceutical Intermediate: A critical building block in the synthesis of active pharmaceutical ingredients (APIs) for potential CNS-targeting drugs.
• Medicinal Chemistry Research: Used in lead optimization and structure-activity relationship (SAR) studies to develop new therapeutic candidates.
• Process Chemistry Development: Employed in route scouting and scale-up processes for the production of novel chemical entities.
• Library Synthesis: Serves as a versatile scaffold for generating diverse compound libraries for high-throughput screening.
• Academic Research: Utilized in university and institutional labs for studying synthetic methodologies and heterocyclic chemistry.
• Contract Research & Manufacturing (CRO/CMO): A key raw material for organizations providing custom synthesis and development services.

Basic Information

Product Name	1-Boc-4-Methyl-4-Morpholin-4-Yl-Piperidine
CAS No.	864369-95-9
Molecular Formula	C15H28N2O3
Molecular Weight	284.40 g/mol
Synonyms	1-Boc-4-Methyl-4-(morpholin-4-yl)piperidine; tert-Butyl 4-methyl-4-morpholinopiperidine-1-carboxylate; 4-Methyl-4-morpholino-1-piperidinecarboxylic Acid 1,1-Dimethylethyl Ester; 1-(tert-Butoxycarbonyl)-4-methyl-4-morpholinopiperidine; 4-Methyl-4-(4-morpholinyl)-1-piperidinecarboxylic Acid tert-Butyl Ester; 864369-95-9; BOC-4-Methyl-4-Morpholinopiperidine
EINECS	Contact for details

Quality Control

Our 1-Boc-4-Methyl-4-Morpholin-4-Yl-Piperidine is manufactured under a quality management system and undergoes rigorous analytical testing to ensure it meets the high standards required for pharmaceutical research. Each batch is accompanied by a comprehensive Certificate of Analysis (COA) detailing purity, identity, and impurity profiles. We are committed to providing materials suitable for use under cGMP guidelines for early-phase development, ensuring reliable performance and supply chain integrity for our global partners.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry, and well-ventilated place at a controlled room temperature (typically 15-25°C). Due to its hygroscopic (moisture-sensitive) nature, the container must be kept tightly sealed and may require storage under an inert atmosphere for long-term preservation. Keep away from incompatible materials.

Specification

Item	Specification
Appearance	White to off-white crystalline powder
Identification (IR)	Conforms to structure
Identification (HPLC)	Retention time matches reference standard
Assay (HPLC)	≥ 98.0%
Related Substances (HPLC)	Any single impurity ≤ 0.5%; Total impurities ≤ 1.0%
Water Content (KF)	≤ 0.5%
Residue on Ignition	≤ 0.1%

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.