Description

Pyrazino[2,1-C][1,4]Oxazine, Octahydro-, (9Ar)- (9Ci) is a high-purity, advanced pharmaceutical intermediate and heterocyclic building block of significant interest in modern synthetic chemistry. Its complex, saturated bicyclic structure makes it a valuable scaffold for the research and development of novel active pharmaceutical ingredients (APIs), particularly in therapeutic areas requiring sophisticated molecular architectures. This compound is primarily utilized by R&D chemists and process development scientists in the pharmaceutical, agrochemical, and fine chemical industries seeking to innovate and optimize synthetic pathways.

Application

• Pharmaceutical Intermediate: Serves as a critical precursor in the synthesis of complex drug candidates, especially those targeting the central nervous system (CNS) and infectious diseases.
• Agrochemical Research: Used as a key building block for developing new generation herbicides, fungicides, and insecticides with novel modes of action.
• Fine Chemical Synthesis: Employed in academic and industrial laboratories for constructing complex heterocyclic compounds for material science and catalysis research.
• Process Chemistry & Scale-up: Provides a defined, high-quality starting material for optimizing synthetic routes from milligram to kilogram scale in pilot plants.
• Chemical Biology Probes: Utilized in the design and synthesis of molecular probes for studying biological pathways and target engagement.

Basic Information

Product Name	Pyrazino[2,1-C][1,4]Oxazine, Octahydro-, (9Ar)- (9Ci)
CAS No.	508241-14-3
Molecular Formula	C6H10N2O
Molecular Weight	126.16 g/mol
Synonyms	Octahydropyrazino[2,1-c][1,4]oxazine; (9ar)-Octahydro-1H-pyrazino[2,1-c][1,4]oxazine; 1,2,3,4,6,7,8,9-Octahydropyrazino[2,1-c][1,4]oxazine; Pyrazinooxazine, octahydro-; Bicyclic Saturated Pyrazino-oxazine; Advanced Heterocyclic Building Block
EINECS	Contact for details

Quality Control

Every batch of Pyrazino[2,1-C][1,4]Oxazine, Octahydro-, (9Ar)- (9Ci) is manufactured under strict quality management systems and undergoes comprehensive analytical characterization to ensure identity, purity, and consistency. Our products are supported by a detailed Certificate of Analysis (COA) that includes data from HPLC, GC, NMR, and mass spectrometry. We are committed to meeting the stringent requirements of cGMP for advanced intermediates and support regulatory filings with complete traceability and documentation.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry, well-ventilated place at controlled room temperature (15-25°C). Keep away from incompatible materials. For long-term storage, consider under an inert atmosphere to maintain optimal purity.

Specification

Item	Specification
Appearance	White to off-white crystalline powder
Identification (IR)	Conforms to reference spectrum
Identification (NMR)	Conforms to structure
Purity (HPLC)	≥ 98.0%
Related Substances (HPLC)	Individual impurity ≤ 0.5%; Total impurities ≤ 2.0%
Residual Solvents (GC)	Complies with ICH Q3C guidelines
Water Content (KF)	≤ 0.5% w/w
Residue on Ignition	≤ 0.1%

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.