Description

Relacatib is a potent and selective cathepsin K inhibitor, a key target for the treatment of bone-related disorders. This high-purity compound is essential for pharmaceutical research and development, offering a critical tool for investigating novel therapeutic pathways. It is primarily utilized by researchers and manufacturers in the pharmaceutical and biotechnology sectors focused on osteoporosis, arthritis, and other conditions involving bone resorption.

Application

• Pharmaceutical R&D: Serves as a reference standard and active pharmaceutical ingredient (API) intermediate in the development of cathepsin K inhibitors.
• Biochemical Research: Used as a selective inhibitor in enzymatic assays to study the role of cathepsin K in bone metabolism and disease pathology.
• Preclinical Studies: Employed in in vitro and in vivo models to evaluate efficacy and pharmacokinetics for potential osteoporosis treatments.
• Chemical Synthesis: Acts as a key building block for the synthesis of more complex therapeutic agents targeting cysteine proteases.

Basic Information

Product Name	Relacatib
CAS No.	362505-84-8
Molecular Formula	C₁₆H₁₈F₃N₃O₃S
Molecular Weight	389.39 g/mol
Synonyms	N-((1S)-2,2,2-Trifluoro-1-{[(2S)-2-(methylamino)-3,3,3-trifluoropropanoyl]amino}ethyl)-1-benzothiophene-2-carboxamide; SB-462795; Relacatib (SB-462795); Cathepsin K Inhibitor IV; SB462795
EINECS	Contact for details

Quality Control

Our Relacatib is manufactured under strict quality management systems. Each batch undergoes comprehensive analytical testing, including HPLC for purity and identity confirmation via spectroscopic methods, to ensure it meets the high standards required for research and development. Certificates of Analysis (COA) with detailed specifications are provided to guarantee batch-to-batch consistency and traceability.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry place at controlled room temperature (15-25°C). This product is hygroscopic (moisture-sensitive) and must be kept under inert conditions or in a desiccator to maintain stability.

Specification

Item	Specification
Appearance	White to off-white solid
Identification (IR)	Conforms to structure
Identification (HPLC)	Conforms to reference
Purity (HPLC)	≥98.0%
Water Content (KF)	≤0.5%
Residue on Ignition	≤0.1%

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.