Description

Tak-071 is a high-purity, non-natural amino acid derivative and advanced pharmaceutical intermediate designed for research and development. This compound is critical for medicinal chemists exploring novel therapeutic agents, particularly in the fields of oncology and neurology. It is primarily utilized by pharmaceutical R&D laboratories, biotechnology firms, and academic research institutions engaged in drug discovery programs.

Application

• Pharmaceutical Intermediate: Serves as a key building block in the synthesis of novel active pharmaceutical ingredients (APIs) for preclinical and clinical studies.
• Medicinal Chemistry Research: Used as a core scaffold or precursor for structure-activity relationship (SAR) studies to optimize drug potency and selectivity.
• Proteolysis-Targeting Chimera (PROTAC) Development: Employed in the design and synthesis of heterobifunctional molecules for targeted protein degradation.
• Peptidomimetic Design: Incorporated into peptide analogs to enhance metabolic stability, bioavailability, and binding affinity.
• Chemical Biology Probes: Utilized to create tool compounds for investigating specific biological pathways and target validation.
• Contract Research & Manufacturing (CRO/CMO): Supplied to service organizations supporting outsourced drug discovery and development projects.

Basic Information

Product Name	Tak-071
CAS No.	1820812-16-5
Molecular Formula	Contact for details
Molecular Weight	Contact for details
Synonyms	TAK-071; TAK071; UNII-9L8K1B8E9F; (2S)-2-Amino-3-[(4-fluorophenyl)methylamino]propanoic acid derivative; GPR52 agonist intermediate; 1820812-16-5; GPR52 modulator precursor
EINECS	Contact for details

Quality Control

Our Tak-071 is manufactured under strict quality management systems to ensure batch-to-batch consistency and high purity for research applications. Quality is verified through comprehensive analytical techniques including HPLC, NMR, and mass spectrometry. A Certificate of Analysis (COA) detailing purity, identity, and impurity profiles is provided with each shipment to support your regulatory and research documentation needs.

Storage

Preserve in a tightly closed container, protected from light. Store at controlled room temperature (15-25°C) in a dry, well-ventilated area. The product is hygroscopic (moisture-sensitive) and should be handled under an inert atmosphere for long-term stability.

Specification

Item	Specification
Appearance	White to off-white solid
Identification (HPLC/MS)	Conforms
Purity (HPLC)	≥ 98.0%
Water Content (KF)	≤ 1.0%
Residue on Ignition	≤ 0.1%

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.