Description

3-[(1-Pyrazin-2-Yl-Ethylamino)-Methyl]-Piperidine-1-Carboxylic Acid tert-Butyl Ester is a high-purity, advanced pharmaceutical intermediate designed for complex organic synthesis. This compound is critical for research and development in medicinal chemistry, particularly in the construction of novel drug candidates. It is primarily utilized by pharmaceutical R&D laboratories and fine chemical manufacturers requiring a reliable, high-quality building block for active pharmaceutical ingredient (API) synthesis.

Application

• Pharmaceutical Intermediate: A key building block in the synthesis of novel drug candidates, particularly in central nervous system (CNS) and other therapeutic areas.
• Medicinal Chemistry Research: Used in structure-activity relationship (SAR) studies and lead optimization for new molecular entities.
• Process Chemistry Development: Serves as a critical intermediate in scaling up synthetic routes from laboratory to pilot plant scale.
• Custom Synthesis: Employed by contract research and manufacturing organizations (CROs/CMOs) for client-specific molecule development.
• Academic Research: Utilized in university and institutional labs for exploring new heterocyclic chemistry and reaction methodologies.
• Library Synthesis: A valuable scaffold for generating diverse compound libraries for high-throughput screening.

Basic Information

Product Name	3-[(1-Pyrazin-2-Yl-Ethylamino)-Methyl]-Piperidine-1-Carboxylic Acid tert-Butyl Ester
CAS No.	1289388-16-4
Molecular Formula	C17H26N4O2
Molecular Weight	318.42 g/mol
Synonyms	1-Boc-3-[(1-(pyrazin-2-yl)ethylamino)methyl]piperidine; tert-Butyl 3-[[[1-(2-pyrazinyl)ethyl]amino]methyl]-1-piperidinecarboxylate; 1-Piperidinecarboxylic acid, 3-[[[1-(2-pyrazinyl)ethyl]amino]methyl]-, 1,1-dimethylethyl ester; 3-[(1-Pyrazin-2-ylethylamino)methyl]piperidine-1-carboxylic acid tert-butyl ester; BOC-protected pyrazinylpiperidine derivative; (3-((1-(Pyrazin-2-yl)ethylamino)methyl)piperidin-1-yl)(tert-butoxy)methanone
EINECS	Contact for details

Quality Control

Our 3-[(1-Pyrazin-2-Yl-Ethylamino)-Methyl]-Piperidine-1-Carboxylic Acid tert-Butyl Ester is manufactured under strict quality management systems. Each batch undergoes rigorous analytical testing, including HPLC, NMR, and mass spectrometry, to ensure identity, purity, and consistency. We provide comprehensive Certificates of Analysis (COA) with each shipment, detailing all specifications and test results. Our quality commitment aligns with cGMP principles for pharmaceutical intermediates.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry, and well-ventilated area at a controlled room temperature (15-25°C). Keep the container tightly sealed when not in use to protect from moisture. For long-term storage, consider storing under an inert atmosphere.

Specification

Item	Specification
Appearance	White to off-white solid
Identification (IR)	Conforms to structure
Identification (NMR)	Conforms to structure
Purity (HPLC)	≥ 97.0%
Water Content (KF)	≤ 0.5%
Residue on Ignition	≤ 0.1%
Heavy Metals	≤ 10 ppm

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.