Description

5-Methyl-6-Morpholinopyridin-3-Ylboronic Acid is a high-purity boronic acid derivative, a critical building block in modern synthetic organic chemistry. Its value lies in enabling efficient carbon-carbon bond formation via the Suzuki-Miyaura cross-coupling reaction, a cornerstone for constructing complex molecular architectures. This compound is essential for researchers and manufacturers in the pharmaceutical and agrochemical industries developing novel active ingredients, as well as in advanced materials science.

Application

• Pharmaceutical Intermediate: A key synthon for constructing pyridine-based scaffolds in drug discovery and development, particularly for kinase inhibitors and other small molecule therapeutics.
• Agrochemical Synthesis: Used in the research and production of advanced crop protection agents and herbicides with complex heterocyclic structures.
• Material Science Research: Serves as a precursor for creating functionalized organic molecules used in organic light-emitting diodes (OLEDs) and electronic materials.
• Chemical Biology Probes: Employed in the synthesis of labeled compounds and molecular probes for studying biological pathways and target engagement.
• Cross-Coupling Reactions: Primarily utilized in palladium-catalyzed Suzuki-Miyaura cross-coupling to introduce the substituted pyridyl moiety into target molecules.
• Library Synthesis: A valuable building block for generating diverse compound libraries in high-throughput screening and medicinal chemistry programs.

Basic Information

Product Name	5-Methyl-6-Morpholinopyridin-3-Ylboronic Acid
CAS No.	1191062-85-7
Molecular Formula	C10H15BN2O3
Molecular Weight	222.05 g/mol
Synonyms	(5-Methyl-6-morpholinopyridin-3-yl)boronic acid; 5-Methyl-6-morpholino-3-pyridineboronic acid; 3-Borono-5-methyl-6-morpholinopyridine; 6-Morpholino-5-methylpyridine-3-boronic acid; Boronic acid, B-(5-methyl-6-morpholino-3-pyridinyl)-; 1191062-85-7
EINECS	Contact for details

Quality Control

Our 5-Methyl-6-Morpholinopyridin-3-Ylboronic Acid is manufactured under strict quality management systems. Each batch undergoes comprehensive analytical testing, including HPLC for purity, NMR for structural confirmation, and Karl Fischer titration for moisture content, to ensure it meets the stringent requirements for advanced synthetic applications. A Certificate of Analysis (COA) detailing all specifications is provided with every shipment.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry, and well-ventilated place at a controlled room temperature (typically 15-25°C). This product is hygroscopic (moisture-sensitive) and must be kept under an inert atmosphere (e.g., nitrogen or argon) for long-term storage to maintain stability and purity.

Specification

Item	Specification
Appearance	White to off-white powder or crystalline solid
Identification (IR)	Conforms to structure
Identification (NMR)	Conforms to structure
Purity (HPLC)	≥95% (Typical 97-99%)
Water Content (KF)	≤1.0%

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.