Tinib Antineoplastic Drugs

Tinib Antineoplastic Drugs

Tinib antineoplastic drugs are a major class of targeted cancer therapies that inhibit dysregulated tyrosine kinases or serine/threonine kinases involved in tumor growth, angiogenesis, and metastasis. Represented by imatinib, erlotinib, gefitinib, sunitinib, sorafenib, and numerous next-generation inhibitors, these APIs block oncogenic signaling pathways such as EGFR, VEGFR, PDGFR, BCR-ABL, ALK, and RET. Their precision targeting enables high efficacy with reduced systemic toxicity compared to traditional chemotherapy. Tinib drugs are widely used in leukemia, lung cancer, renal cancer, gastrointestinal stromal tumors, and melanoma. Resistance caused by kinase mutations has led to the development of multi-targeted and mutation-specific inhibitors, making tinibs a cornerstone of precision oncology.

1-[4-(4-Aminofuro[2,3-D]Pyrimidin-5-Yl)Phenyl]-3-[2-Fluoro-5-(Trifluoromethyl)Phenyl]Urea CAS NO 501693-48-7

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CAS No.:501693-48-7

Grade:Pharmacy Grade

Content:99.90%

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Cp-724714 CAS NO 537705-08-1

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CAS No.:537705-08-1

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Content:99.90%

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Taz-204 CAS NO 539854-53-0

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CAS No.:539854-53-0

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Content:99.90%

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Cdk4 Inhibitor CAS NO 546102-60-7

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CAS No.:546102-60-7

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Content:99.90%

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Litronesib (Racemate) CAS NO 546111-97-1

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CAS No.:546111-97-1

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Content:99.90%

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Cedirannib CAS NO 557795-03-6

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CAS No.:557795-03-6

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Content:99.90%

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Sunitinib CAS NO 557795-19-4

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CAS No.:557795-19-4

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Content:99.90%

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n-{3-[(4-Ethylphenyl)Amino]Quinoxalin-2-Yl}-4-Fluorobenzenesulfonamide CAS NO 577960-49-7

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CAS No.:577960-49-7

Grade:Pharmacy Grade

Content:99.90%

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