Description

4-Methoxy-2-Methyl-5-Azaindole is a high-purity, advanced pharmaceutical intermediate belonging to the azaindole class of heterocyclic compounds. This specialized building block is critical for the synthesis of novel, small-molecule drug candidates, particularly in oncology and antiviral research. It is primarily utilized by pharmaceutical R&D departments and fine chemical manufacturers engaged in developing targeted therapies.

Application

• Pharmaceutical Intermediate: A key synthon for the research and development of kinase inhibitors and other targeted therapeutic agents.
• Oncology Drug Discovery: Serves as a core scaffold in the synthesis of compounds targeting specific cancer pathways.
• Antiviral Agent Synthesis: Used in the construction of molecules with potential activity against various viral targets.
• Chemical Biology & Proteomics: Employed as a molecular probe or tag in studying protein-ligand interactions and cellular processes.
• Agrochemical Research: Potential intermediate for developing new generation pesticides and plant growth regulators.
• Material Science: Exploration of its use in organic electronic materials due to its heterocyclic, electron-rich structure.

Basic Information

Product Name	4-Methoxy-2-Methyl-5-Azaindole
CAS No.	936572-00-8
Molecular Formula	C9H10N2O
Molecular Weight	162.19 g/mol
Synonyms	5-Azaindole, 4-methoxy-2-methyl-; 2-Methyl-4-methoxy-1H-pyrrolo[3,2-b]pyridine; 4-Methoxy-2-methyl-1H-pyrrolo[3,2-b]pyridine; 1H-Pyrrolo[3,2-b]pyridine, 4-methoxy-2-methyl-; 2-Methyl-4-methoxy-5-azaindole; 4-Methoxy-2-methyl-7-azaindole (common misnomer); 936572-00-8
EINECS	Contact for details

Quality Control

Our 4-Methoxy-2-Methyl-5-Azaindole is manufactured under strict quality management systems. Each batch undergoes rigorous analytical testing, including HPLC, NMR, and MS, to ensure identity, purity, and consistency. We provide comprehensive Certificates of Analysis (COA) with every shipment, detailing all specifications and test results. Our quality commitment supports compliance with cGMP and ICH guidelines for pharmaceutical intermediates.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry, and well-ventilated place at a controlled room temperature (15-25°C). Keep the container tightly sealed in a dry environment to minimize moisture uptake.

Specification

Item	Specification
Appearance	White to off-white powder
Identification (IR)	Conforms to structure
Identification (HPLC)	Conforms to reference
Purity (HPLC)	≥ 98.0%
Water Content (KF)	≤ 0.5%
Residue on Ignition	≤ 0.1%
Heavy Metals	≤ 10 ppm

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.