Description

3-Bromo-5,6-Dimethoxy-4-Azaindole is a high-purity, advanced pharmaceutical intermediate characterized by its unique azaindole scaffold. This compound matters as a critical building block in modern medicinal chemistry, enabling the synthesis of novel drug candidates with targeted biological activity. It is primarily needed by research and development teams in the pharmaceutical and biotechnology sectors for the development of new therapeutic agents.

Application

• Pharmaceutical Intermediate: A key synthon for the research and development of new active pharmaceutical ingredients (APIs), particularly in kinase inhibitor programs.
• Medicinal Chemistry Research: Used as a versatile scaffold for structure-activity relationship (SAR) studies and lead optimization in drug discovery.
• Biochemical Tool Compound: Serves as a precursor for labeled probes or inhibitors used in biochemical and cellular assays to study disease pathways.
• Contract Manufacturing: Supplied to CDMOs (Contract Development and Manufacturing Organizations) for custom synthesis and scale-up projects.
• Academic Research: Utilized in university and institutional labs for exploratory synthetic chemistry and novel heterocycle development.

Basic Information

Product Name	3-Bromo-5,6-Dimethoxy-4-Azaindole
CAS No.	882033-34-3
Molecular Formula	C9H9BrN2O2
Molecular Weight	257.09 g/mol
Synonyms	3-Bromo-5,6-dimethoxy-1H-pyrrolo[3,2-c]pyridine; 4-Azaindole, 3-bromo-5,6-dimethoxy-; 1H-Pyrrolo[3,2-c]pyridine, 3-bromo-5,6-dimethoxy-; 5,6-Dimethoxy-3-bromo-4-azaindole; 3-Bromo-5,6-dimethoxy-4-aza-indole; 882033-34-3; 3-Br-5,6-(OMe)2-4-azaindole
EINECS	Contact for details

Quality Control

Our 3-Bromo-5,6-Dimethoxy-4-Azaindole is manufactured under strict quality management systems. Each batch undergoes rigorous analytical testing, including HPLC, NMR, and mass spectrometry, to ensure identity, purity, and consistency. We provide comprehensive Certificates of Analysis (COA) with every shipment, detailing all specifications and test results. Our quality commitment aligns with cGMP principles for pharmaceutical intermediates, ensuring reliability for your critical R&D and scale-up processes.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry, and well-ventilated place at a controlled room temperature (typically 15-25°C). Keep the container sealed to protect this light-sensitive material from moisture and atmospheric contamination.

Specification

Item	Specification
Appearance	White to off-white powder
Identification (IR)	Conforms to structure
Identification (HPLC)	Conforms to reference standard
Purity (HPLC)	≥ 98.0%
Water Content (KF)	≤ 0.5%
Residue on Ignition	≤ 0.1%
Heavy Metals	≤ 20 ppm

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.