Description

(5Alpha,6Alpha)-7,8-Didehydro-4,5-Epoxy-3-Methoxy-17-Methylmorphinan-6-Yl (1S)-7,7-Dimethyl-2-Oxobicyclo[2.2.1]Heptane-1-Methanesulphonate CAS NO 83968-47-2 is a high-purity, specialized chemical intermediate with a complex molecular architecture. This compound is of significant value for its role in advanced pharmaceutical synthesis and research, particularly in the development of novel therapeutic agents. It is primarily needed by research institutions, pharmaceutical R&D laboratories, and fine chemical manufacturers focused on opioid receptor-targeted molecules and complex organic synthesis.

Application

• Pharmaceutical Intermediate: Critical building block in the research and synthesis of novel opioid analgesics and related receptor modulators.
• Medicinal Chemistry Research: Used as a key precursor or reference standard in structure-activity relationship (SAR) studies for central nervous system (CNS) active compounds.
• Process Development: Serves as a high-value intermediate in the scale-up and optimization of synthetic routes for complex active pharmaceutical ingredients (APIs).
• Analytical Reference Standard: Employed in analytical method development and validation (e.g., HPLC, LC-MS) for quality control and impurity profiling in pharmaceutical manufacturing.
• Biochemical Research: Utilized in in-vitro studies to investigate binding affinity and pharmacological activity at specific receptor sites.
• Custom Synthesis: A starting material for the custom synthesis of derivatives and analogs for proprietary drug discovery programs.

Basic Information

Product Name	(5Alpha,6Alpha)-7,8-Didehydro-4,5-Epoxy-3-Methoxy-17-Methylmorphinan-6-Yl (1S)-7,7-Dimethyl-2-Oxobicyclo[2.2.1]Heptane-1-Methanesulphonate
CAS No.	83968-47-2
Molecular Formula	C28H37NO6S
Molecular Weight	515.66 g/mol
Synonyms	Oxycodone Camphorsulfonate; Oxycodone (+)-Camphor-10-sulfonate Salt; 14-Hydroxydihydrocodeinone Camphorsulfonate; (5α,6α)-7,8-Didehydro-4,5-epoxy-3-methoxy-17-methylmorphinan-6-yl (1S)-7,7-dimethyl-2-oxobicyclo[2.2.1]heptane-1-methanesulfonate; Oxycodone D-Camphorsulfonate; Oxycodone-(+)-10-camphorsulfonic acid salt
EINECS	Contact for details

Quality Control

Our production of this high-purity intermediate adheres to strict quality management systems. Every batch undergoes comprehensive analytical testing, including HPLC for purity and chiral integrity, to ensure it meets the exacting standards required for pharmaceutical research and development. A detailed Certificate of Analysis (COA) is provided with each shipment, documenting identity, assay, impurity profile, and other critical parameters.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry place at controlled room temperature (15-25°C). Due to its hygroscopic (moisture-sensitive) nature, the container must be kept tightly sealed in a dry environment to prevent degradation. For long-term storage, consider desiccants or an inert atmosphere.

Specification

Item	Specification
Appearance	White to off-white crystalline powder
Identification (IR)	Conforms to reference spectrum
Identification (HPLC)	Retention time matches reference standard
Assay (HPLC)	≥ 98.0%
Chiral Purity	≥ 99.0%
Water Content (KF)	≤ 1.0%
Residue on Ignition	≤ 0.1%
Heavy Metals	≤ 20 ppm
Related Substances (HPLC)	Individual impurity ≤ 0.5%, Total impurities ≤ 1.5%

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.