Description

Amperozide is a potent and selective 5-HT2A receptor antagonist with significant pharmacological activity. This compound is of primary interest for its role in advanced neuropharmacological research and as a key intermediate in the development of novel therapeutic agents. It is essential for researchers and manufacturers in the pharmaceutical and life science sectors focused on central nervous system disorders.

Application

• Neuropharmacological Research: A critical reference standard and tool compound for studying serotonin (5-HT2A) receptor function and signaling pathways.
• Drug Discovery & Development: Serves as a high-purity chemical building block or intermediate in the synthesis of potential antipsychotic and anxiolytic drug candidates.
• Biochemical Assays: Used in in vitro binding and functional assays to screen for receptor activity and evaluate compound libraries.
• Academic & Institutional Research: Supports fundamental neuroscience studies in universities and research institutes investigating behavior, cognition, and neuropsychiatric conditions.
• Preclinical Studies: Employed in animal model research to understand the pharmacokinetics and pharmacodynamics of 5-HT2A antagonism.

Basic Information

Product Name	Amperozide
CAS No.	75558-90-6
Molecular Formula	C23H32FN3O
Molecular Weight	385.52 g/mol
Synonyms	4'-Fluoro-4-[4-(2-pyridinyl)-1-piperazinyl]butyrophenone; FG 5606; FG-5606; Amperozide hydrochloride (salt form); N-(4-Fluorophenyl)-4-(4-pyridin-2-ylpiperazin-1-yl)butan-1-one
EINECS	Contact for details

Quality Control

Our Amperozide is manufactured under strict quality management systems. Each batch undergoes rigorous analytical testing, including HPLC for purity and identity confirmation via IR and MS, to ensure it meets the high standards required for research applications. A comprehensive Certificate of Analysis (COA) detailing all specifications is provided with every shipment.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry place at controlled room temperature (15-25°C). The compound is light-sensitive and should be handled under appropriate conditions to maintain stability.

Specification

Item	Specification
Appearance	White to off-white powder
Identification (IR)	Conforms to reference spectrum
Identification (HPLC)	Retention time matches reference standard
Purity (HPLC)	≥ 98.0%
Related Substances (HPLC)	Total impurities ≤ 2.0%
Water Content (KF)	≤ 0.5%
Residue on Ignition	≤ 0.1%

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.