Description

Flupirtine Maleate is a centrally acting, non-opioid analgesic agent with muscle relaxant properties. This compound is valued for its unique mechanism of action, acting as a selective neuronal potassium channel opener, which differentiates it from NSAIDs and opioids. It is primarily utilized in the pharmaceutical industry for the research, development, and production of prescription medications targeting acute and chronic pain management, including conditions like fibromyalgia and tension headaches.

Application

• Pharmaceutical Active Ingredient (API): Core component in the formulation of prescription analgesic medications.
• Neurological Pain Research: A key compound in preclinical and clinical studies investigating non-opioid pathways for pain relief.
• Muscle Relaxant Formulations: Used in developing drugs aimed at alleviating muscle tension and spasticity associated with pain.
• Reference Standard: Serves as a high-purity standard in analytical laboratories for quality control and method development.
• Drug Development Intermediates: Employed in the synthetic pathways for creating novel analgesic derivatives.

Basic Information

Product Name	Flupirtine Maleate
CAS No.	75507-68-5
Molecular Formula	C15H17FN4O2 • C4H4O4
Molecular Weight	424.39 g/mol
Synonyms	Ethyl {2-Amino-6-[(4-fluorophenyl)methylamino]-3-pyridinyl}carbamate Maleate; D 9998; Katadolon; Trancolong; E-371; Flupirtin Maleate; Flupirtine Hydrogen Maleate; (±)-Flupirtine Maleate
EINECS	Contact for details

Quality Control

Our Flupirtine Maleate is manufactured under strict quality management systems. Each batch undergoes comprehensive analytical testing to ensure it meets high-purity standards suitable for pharmaceutical research and development. Certificates of Analysis (COA) detailing purity, identity, and impurity profiles are available upon request.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry place at controlled room temperature (15-25°C). Due to its hygroscopic nature, the container must be kept tightly sealed in a dry environment to prevent moisture absorption.

Specification

Item	Specification
Appearance	White to off-white crystalline powder
Identification (IR)	Conforms to reference spectrum
Identification (HPLC)	Retention time corresponds to reference standard
Assay (HPLC)	≥98.5%
Related Substances (HPLC)	Total impurities ≤1.5%
Single Maximum Impurity	≤0.5%
Loss on Drying	≤0.5%
Residue on Ignition	≤0.1%
Heavy Metals	≤20 ppm

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.