Description

4-Thiazolidinecarboxylic Acid, 5,5-Dimethyl-2-[[(2-Phenylacetyl)Amino]Methyl]-, (2R,4S)- is a high-purity, stereochemically defined thiazolidine derivative of significant interest in advanced pharmaceutical research and development. Its core value lies in its role as a sophisticated chiral building block and potential pharmacophore for designing novel therapeutic agents. This compound is essential for researchers and manufacturers in the pharmaceutical and biotechnology sectors, particularly those focused on developing enzyme inhibitors, prodrugs, and targeted small molecule therapies.

Application

• Pharmaceutical Intermediate: Serves as a critical chiral synthon in the multi-step synthesis of complex drug candidates.
• Enzyme Inhibitor Research: Used in the design and development of potential inhibitors for metalloproteases and other enzyme targets due to its thiazolidine core.
• Prodrug Development: Investigated as a potential carrier moiety in prodrug strategies to improve drug solubility, stability, or targeted delivery.
• Chemical Biology Probes: Employed in the creation of molecular probes to study biological pathways and protein function.
• Peptidomimetics: Acts as a conformationally constrained scaffold in the design of peptidomimetic compounds with enhanced metabolic stability.
• Asymmetric Synthesis: Utilized as a chiral auxiliary or reagent in stereoselective synthetic transformations.

Basic Information

Item	Details
Product Name	4-Thiazolidinecarboxylic Acid, 5,5-Dimethyl-2-[[(2-Phenylacetyl)Amino]Methyl]-, (2R,4S)-
CAS No.	73184-06-2
Molecular Formula	C15H20N2O3S
Molecular Weight	308.40 g/mol
Synonyms	(2R,4S)-5,5-Dimethyl-2-[(2-phenylacetamido)methyl]thiazolidine-4-carboxylic acid; (4S)-5,5-Dimethyl-2-[[(2-phenylacetyl)amino]methyl]-4-thiazolidinecarboxylic acid (2R); D-Penicillamine derivative; Thiazolidine-4-carboxylic acid derivative; Chiral thiazolidine; N-(Phenylacetyl)-D-penicillamine thiazolidine derivative
EINECS	Contact for details

Quality Control

Our 4-Thiazolidinecarboxylic Acid derivative is manufactured under strict quality management systems. Each batch undergoes comprehensive analytical testing, including chiral purity verification by HPLC, to ensure it meets the stringent requirements for pharmaceutical R&D. A detailed Certificate of Analysis (COA) documenting identity, purity, and chiral integrity is provided with every shipment.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry place at a controlled room temperature (15-25°C). This product is hygroscopic (moisture-sensitive) and must be kept under anhydrous conditions. For long-term storage, consider storing under an inert atmosphere.

Specification

Item	Specification
Appearance	White to off-white powder
Identification (IR)	Conforms to structure
Assay (HPLC)	≥ 98.0%
Chiral Purity (HPLC)	≥ 99.0% de
Water Content (KF)	≤ 1.0%
Residue on Ignition	≤ 0.1%
Heavy Metals	≤ 10 ppm

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.