Description

5H-1,2,4-Triazino[5,6-B]Indole,5,8-Dimethyl-3-[[2-(4-Morpholinyl)Ethyl]Thio]-(9Ci) is a sophisticated heterocyclic organic compound that serves as a critical advanced pharmaceutical intermediate and research chemical. Its unique molecular architecture, featuring fused triazine and indole rings with a morpholinoethylthio side chain, makes it a valuable scaffold for medicinal chemistry and drug discovery programs. This compound is primarily utilized by pharmaceutical R&D teams and contract research organizations (CROs) focused on developing novel therapeutic agents.

Application

• Pharmaceutical Intermediate: Key building block in the synthesis of novel drug candidates targeting various disease pathways.
• Medicinal Chemistry Research: Core scaffold for structure-activity relationship (SAR) studies and lead optimization in drug discovery.
• Biochemical Probe Development: Used to create tools for studying enzyme inhibition and receptor-ligand interactions in biological systems.
• Academic Research: Employed in university and institutional labs for investigating heterocyclic chemistry and new synthetic methodologies.
• High-Throughput Screening (HTS): Component of specialized compound libraries screened for biological activity against novel targets.
• Preclinical Development: Serves as a precursor in the development of active pharmaceutical ingredients (APIs) for preclinical testing.

Basic Information

Product Name	5H-1,2,4-Triazino[5,6-B]Indole,5,8-Dimethyl-3-[[2-(4-Morpholinyl)Ethyl]Thio]-(9Ci)
CAS No.	603946-36-7
Molecular Formula	C17H21N5OS
Molecular Weight	343.45 g/mol
Synonyms	5,8-Dimethyl-3-((2-morpholinoethyl)thio)-5H-[1,2,4]triazino[5,6-b]indole; 3-[(2-Morpholin-4-ylethyl)sulfanyl]-5,8-dimethyl-5H-[1,2,4]triazino[5,6-b]indole; 5H-[1,2,4]Triazino[5,6-b]indole, 5,8-dimethyl-3-[[2-(4-morpholinyl)ethyl]thio]-; 603946-36-7; 5,8-Dimethyl-3-((2-morpholinoethyl)thio)-5H-1,2,4-triazino[5,6-b]indole
EINECS	Contact for details

Quality Control

Our production of this high-value intermediate adheres to strict quality management systems. Every batch is characterized and tested using advanced analytical techniques including HPLC, NMR, and mass spectrometry to ensure identity, purity, and consistency. A comprehensive Certificate of Analysis (COA) detailing all specifications is provided with each shipment. We support cGMP-compliant manufacturing for advanced pharmaceutical applications upon request.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry, and well-ventilated area at a controlled room temperature (typically 15-25°C). The compound may be light-sensitive and should be handled under appropriate conditions to maintain stability.

Specification

Item	Specification
Appearance	Off-white to light yellow solid
Identification (IR)	Conforms to structure
Identification (NMR)	Conforms to structure
Purity (HPLC)	≥ 97.0%
Related Substances (HPLC)	Total impurities ≤ 3.0%
Residual Solvents (GC)	Meets ICH guidelines
Loss on Drying	≤ 0.5%

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.