Description

(5-Bromo-1-Benzothiophen-2-Yl)(Morpholino)Methanone is a high-purity, advanced pharmaceutical intermediate characterized by its distinct benzothiophene core functionalized with bromine and a morpholino carbonyl group. This compound is critical for medicinal chemistry research and development, serving as a versatile building block for the synthesis of novel bioactive molecules. It is primarily utilized by R&D chemists and process development scientists in the pharmaceutical and agrochemical industries to create new drug candidates and active ingredients.

Application

• Pharmaceutical Intermediate: A key precursor in the synthesis of potential therapeutic agents, particularly those targeting kinase inhibition or other enzyme-related pathways.
• Medicinal Chemistry Research: Used as a core scaffold or derivatization point for structure-activity relationship (SAR) studies and lead optimization in drug discovery programs.
• Agrochemical Development: Serves as a building block for creating novel active ingredients in crop protection and pesticide formulations.
• Chemical Biology Probes: Utilized in the development of molecular probes for studying biological processes and target validation.
• Organic Synthesis: Employed in advanced organic synthesis for constructing complex heterocyclic systems due to its reactive bromine substituent.

Basic Information

Product Name	(5-Bromo-1-Benzothiophen-2-Yl)(Morpholino)Methanone
CAS No.	439107-98-9
Molecular Formula	C₁₃H₁₂BrNO₂S
Molecular Weight	326.21 g/mol
Synonyms	5-Bromo-1-benzothiophen-2-yl morpholin-4-yl methanone; 5-Bromo-1-benzothiophene-2-carboxylic acid morpholide; Morpholine, 4-[(5-bromo-2-benzothienyl)carbonyl]-; (5-Bromobenzo[b]thiophen-2-yl)(morpholino)methanone; 439107-98-9; 5-Bromo-N-morpholinobenzo[b]thiophene-2-carboxamide
EINECS	Contact for details

Quality Control

Our (5-Bromo-1-Benzothiophen-2-Yl)(Morpholino)Methanone is manufactured under strict quality management systems. Each batch undergoes rigorous analytical testing, including HPLC, NMR, and mass spectrometry, to ensure identity, purity, and consistency. We provide comprehensive Certificates of Analysis (COA) with each shipment, detailing all critical quality attributes. Our commitment to quality supports your R&D and scale-up activities with reliable, traceable materials.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry, well-ventilated area at a controlled room temperature (15-25°C). Keep the container tightly sealed to protect from moisture. For long-term storage, consider storing under an inert atmosphere.

Specification

Item	Specification
Appearance	White to off-white crystalline powder
Identification (IR)	Conforms to structure
Identification (HPLC)	Conforms to reference standard
Purity (HPLC)	≥ 97.0%
Water Content (KF)	≤ 0.5%
Residue on Ignition	≤ 0.1%
Heavy Metals	≤ 20 ppm

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.