Description

5-Formyl-2-(2-Morpholinoethoxy)Phenylboronic Acid is a sophisticated bifunctional organic building block designed for advanced synthetic chemistry. This compound is valued for its dual reactivity, combining a formyl group and a boronic acid moiety, which facilitates efficient cross-coupling and subsequent functionalization in a single molecule. It is primarily utilized by research chemists and process development scientists in the pharmaceutical and agrochemical industries for constructing complex molecular architectures, such as active pharmaceutical ingredients (APIs) and novel bioactive compounds.

Application

• Pharmaceutical Intermediate: A key precursor in the synthesis of complex drug candidates, particularly those requiring Suzuki-Miyaura cross-coupling reactions.
• Agrochemical Research: Used to develop novel active ingredients for crop protection products through modular synthesis.
• Material Science: Serves as a monomer or linker in the creation of functional polymers and organic electronic materials.
• Chemical Biology: Employed in the development of probes and bioconjugates due to its orthogonal reactive handles.
• Catalyst Ligand Synthesis: Acts as a starting material for constructing novel ligand frameworks in transition metal catalysis.
• Library Synthesis: Enables rapid generation of diverse compound libraries for high-throughput screening in drug discovery.

Basic Information

Product Name	5-Formyl-2-(2-Morpholinoethoxy)Phenylboronic Acid
CAS No.	2377611-16-8
Molecular Formula	C₁₃H₁₈BNO₅
Molecular Weight	279.10 g/mol
Synonyms	[2-(2-Morpholin-4-ylethoxy)-5-formylphenyl]boronic acid; 5-Formyl-2-(2-morpholinoethoxy)benzeneboronic acid; 2-(2-Morpholinoethoxy)-5-formylphenylboronic Acid; (5-Formyl-2-(2-morpholinoethoxy)phenyl)boronic acid; Boronic acid, B-[5-formyl-2-[2-(4-morpholinyl)ethoxy]phenyl]-; CAS 2377611-16-8
EINECS	Contact for details

Quality Control

Our 5-Formyl-2-(2-Morpholinoethoxy)Phenylboronic Acid is manufactured under strict quality management systems. Each batch undergoes rigorous analytical testing, including HPLC, NMR, and mass spectrometry, to ensure high purity and consistent performance. Certificates of Analysis (COA) detailing identity, purity, and impurity profiles are provided with every shipment to support your quality assurance and regulatory documentation needs.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry, and well-ventilated place at a controlled room temperature (15-25°C). Due to its hygroscopic nature, the container must be kept tightly sealed under an inert atmosphere (e.g., nitrogen or argon) after opening to prevent moisture absorption and degradation.

Specification

Item	Specification
Appearance	White to off-white powder
Identification (IR)	Conforms to structure
Identification (NMR)	Conforms to structure
Purity (HPLC)	≥ 95.0%
Water Content (KF)	≤ 1.0%

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.