Description

2-Methoxycarbonylindole-5-Boronicacid is a high-value, multi-functional boronic acid derivative and a key synthetic intermediate in modern organic chemistry. Its core value lies in enabling precise carbon-carbon bond formation via Suzuki-Miyaura cross-coupling reactions, a cornerstone of complex molecule assembly. This compound is essential for researchers and manufacturers in the pharmaceutical and agrochemical industries developing novel active ingredients, particularly for constructing indole-based scaffolds.

Application

• Pharmaceutical Intermediate: Critical building block for the synthesis of novel drug candidates, especially those containing functionalized indole cores for oncology, CNS, and anti-inflammatory applications.
• Agrochemical Research: Used in creating advanced active ingredients for crop protection products, leveraging the indole structure for biological activity.
• Material Science: Serves as a monomer or precursor for constructing organic electronic materials, such as OLEDs and conductive polymers.
• Chemical Biology & Proteomics: Employed in the development of enzyme inhibitors, molecular probes, and bioconjugation reagents due to its specific reactivity.
• Academic & R&D Laboratories: A versatile reagent for methodological development in synthetic organic chemistry and catalysis studies.
• Custom Synthesis & Contract Manufacturing: A requested intermediate for the bespoke production of complex molecules for various industrial clients.

Basic Information

Product Name	2-Methoxycarbonylindole-5-Boronicacid
CAS No.	284660-86-2
Molecular Formula	C10H10BNO4
Molecular Weight	219.00 g/mol
Synonyms	5-Borono-1H-indole-2-carboxylic acid methyl ester; Methyl 5-borono-1H-indole-2-carboxylate; 1H-Indole-2-carboxylic acid, 5-borono-, methyl ester; 2-Carbomethoxyindole-5-boronic acid; Methyl 5-boronindole-2-carboxylate; 5-Boron-1H-indole-2-carboxylic acid methyl ester; (2-Methoxycarbonyl-1H-indol-5-yl)boronic acid
EINECS	Contact for details

Quality Control

Our 2-Methoxycarbonylindole-5-Boronicacid is produced under strict quality management protocols to ensure batch-to-batch consistency and high purity, suitable for demanding R&D and scale-up applications. Each lot is accompanied by a comprehensive Certificate of Analysis (COA) detailing purity, identity, and impurity profiles, typically determined by advanced analytical techniques including HPLC, NMR, and IR spectroscopy. We adhere to relevant cGMP and ISO 9001 standards where applicable to guarantee traceability and reliability for our global B2B clients.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry, and well-ventilated place at a controlled room temperature (15-25°C). Due to its hygroscopic (moisture-sensitive) nature, the container must be kept sealed under an inert atmosphere (e.g., nitrogen or argon) after opening to prevent degradation. Keep away from incompatible materials.

Specification

Item	Specification
Appearance	White to off-white powder
Identification (IR)	Conforms to structure
Identification (NMR)	Conforms to structure
Purity (HPLC)	≥ 97.0%
Water Content (KF)	≤ 0.5%
Heavy Metals	≤ 20 ppm

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.